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Legal status
Patent lapsed (non-payment of fees)
| (51) | INT.CL.: (2006.01) |
A61K 31/00 A61K 31/185 A61K 31/357 A61K 31/415 A61K 31/4164 A61K 31/505 A61P 19/00 C07C 45/00 C07C 49/00 C07C 281/00 C07C 337/00 C07D 233/00 C07D 239/00 C07D 317/00 |
| (11) | Number of the document | 4535 |
| (13) | Kind of document | B |
| (21) | Application number | 98-145 |
| (22) | Date of filing the application | 1998-10-15 |
| (41) | Date of publication of the application | 1999-03-25 |
| (45) | Date of publication of patent | 1999-08-25 |
| (86) | Number | PCT/FR97/00487 |
| Date | 1997-03-20 |
| (87) | Number | WO 97/34865 |
| Date | 1997-09-25 |
| (30) | Number | Date | Country code |
| 96/03437 | 1996-03-20 | FR |
| (71) |
HOECHST MARION ROUSSEL,
1 Terrasse Bellini, F-92800 Puteaux,
FR
GENENTECH, INC., 460 Point San Bruno Boulevard, South San Francisco, CA 94080-4990, US |
| (72) |
Serge BERNARD, FR
Denis CARNIATO, FR Jean Francois GOURVEST, FR Jean Georges TEUTSCH, FR Jochen KNOLLE, DE Hans Ulrich STILZ, DE Volkmar WEHNER, DE Sarah C. BODARY, US Thomas R. GADEK, US Robert S. MCDOWELL, US Robert M. PITTI, US |
| (73) |
GENENTECH, INC.,
460 Point San Bruno Boulevard, South San Francisco, CA 94080-4990,
US
AVENTIS PHARMA S.A., 20, Avenue Raymond Aron, 92160 Antony, FR |
| (74) |
Reda ŽABOLIENĖ,
METIDA, Verslo centras "VERTAS", Gynėjų g. 16, LT-01109 Vilnius,
LT
|
| (54) | TRICYCLIC COMPOUNDS HAVING ACTIVITY SPECIFIC FOR INTEGRINS, PARTICULARY ALPHA-GAMA-BETA-3 INTEGRINS, METHOD FOR PREPARING SAME, INTERMEDIATES THEREFOR, USE OF SAID COMPOUNDS AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
| Payment date | Validity (years) | Amount | |
| 2003-03-13 | 7 | 560.00 LTL |
| Patent lapsed (non-payment of fees) | ||
| Invalidation date | 2004-03-20 |