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LT - Tret-butilo (E)-(6-{2[-4-(4-fluorfenil)-6-izopropil-2-[N-metil-N-metilsulfonil)amino] pirimidin-5-il]vinil}-(4R,6S)-2,2-dimetil-[1,3]dioksan-4-il)acetato gamybos būdas
EN - PROCESS FOR THE PRODUCTION OF TERT-BUTYL (E)-(6-{2-[4-(4-FLUOROPHENYL)-6-ISOPROPYL-2-[N-METHYL-N-METHYLSULFONYL)AMINO]PYRIMIDIN-5-YL]VINYL}-(4R,6S)-2,2-DIMETHYL-[1,3]DIOXAN-4-YL)ACETATE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 405/06 (2006.01)
European patent
(11) Number of the document 1155015
(13) Kind of document T
(96) European patent application number 00903810.0
Date of filing the European patent application 2000-02-15
(97) Date of publication of the European application 2001-11-21
(45) Date of publication and mention of the grant of the patent 2008-11-26
(46) Date of publication of the claims translation 2009-03-25
PCT application
(86) Number PCT/GB2000/000481
Date 2000-02-15
PCT application publication
(87) Number WO 2000/049014
Date 2000-08-24
Priority applications
(30) Number Date Country code
9903472 1999-02-17 GB
Inventors
(72)
KOIKE, Haruo, JP
KABAKI, Mikio, JP
TAYLOR, Nigel, Philip, GB
DIORAZIO, Louis, Joseph, GB
Grantee
(73) SHIONOGI & CO., LTD., 1-8, Doshomachi 3-chome, Chuo-ku, Osaka-shi, Osaka 541-0045, JP
AstraZeneca AB, 151 85 Södertälje, SE
Attorney or representative
(74) Liudmila GERASIMOVIČ, IĮ "Liudmila Gerasimovič, Patentinis patikėtinis", Vingrių g. 13-42, LT-01141 Vilnius, LT
Title
(54) Tret-butilo (E)-(6-{2[-4-(4-fluorfenil)-6-izopropil-2-[N-metil-N-metilsulfonil)amino] pirimidin-5-il]vinil}-(4R,6S)-2,2-dimetil-[1,3]dioksan-4-il)acetato gamybos būdas
  PROCESS FOR THE PRODUCTION OF TERT-BUTYL (E)-(6-{2-[4-(4-FLUOROPHENYL)-6-ISOPROPYL-2-[N-METHYL-N-METHYLSULFONYL)AMINO]PYRIMIDIN-5-YL]VINYL}-(4R,6S)-2,2-DIMETHYL-[1,3]DIOXAN-4-YL)ACETATE
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2019-01-28 20 347.00 EUR