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LT - VERFAHREN ZUR HERSTELLUNG VON EPINASTINE-HYDROCHLORID IN DER HOCHSCHMELZENDEN KRISTALLMODIFIKATION
EN - METHOD FOR PRODUCING EPINASTINE HYDROCHLORIDE IN THE HIGH-MELTING CRYSTAL MODIFICATION

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/55 (2006.01)
A61P 37/00 (2006.01)
A61P 37/08 (2006.01)
A61P 43/00 (2006.01)
C07D 487/04 (2006.01)
European patent
(11) Number of the document 1237892
(13) Kind of document T
(96) European patent application number 00985110.6
Date of filing the European patent application 2000-11-29
(97) Date of publication of the European application 2002-09-11
(45) Date of publication and mention of the grant of the patent 2003-04-23
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP0011/942
Date 2000-11-29
PCT application publication
(87) Number WO 0104/0229
Date 2001-06-07
Priority applications
(30) Number Date Country code
19958460 1999-12-03 DE
Inventors
(72)
DACH, Rolf, DE
Grantee
(73) Boehringer Ingelheim Pharma GmbH & Co.KG, Binger Strasse 173, 55218 Ingelheim am Rhein, DE
Title
(54) VERFAHREN ZUR HERSTELLUNG VON EPINASTINE-HYDROCHLORID IN DER HOCHSCHMELZENDEN KRISTALLMODIFIKATION
  METHOD FOR PRODUCING EPINASTINE HYDROCHLORIDE IN THE HIGH-MELTING CRYSTAL MODIFICATION