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LT - IMPROVED PROCESS FOR THE PREPARATION OF WATER-SOLUBLE O-PHOSPHONOOXYMETHYL PRODRUGS
EN - IMPROVED PROCESS FOR THE PREPARATION OF WATER-SOLUBLE O-PHOSPHONOOXYMETHYL PRODRUGS

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 277/22
C07D 249/08
C07D 417/08
European patent
(11) Number of the document 1345915
(13) Kind of document T
(96) European patent application number 01981688.3
Date of filing the European patent application 2001-10-18
(97) Date of publication of the European application 2003-09-24
(45) Date of publication and mention of the grant of the patent 2007-01-31
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2001/032382
Date 2001-10-18
PCT application publication
(87) Number WO 2002/042283
Date 2002-05-30
Priority applications
(30) Number Date Country code
252001 P 2000-11-20 US
Inventors
(72)
CHEN, Chung-Pin, US
CONNOLLY, Timothy Paul, US
KOLLA, Laxma, Reddy, US
MATISKELLA, John, D., US
MUELLER, Richard, H., US
PENDRI, Yadagiri, US
PETSCH, Dejah, T., US
Grantee
(73) Eisai R&D Management Co., Ltd., 6-10, Koishikawa 4-chome, Bunkyo-ku, Tokyo 112-8088, JP
Title
(54) IMPROVED PROCESS FOR THE PREPARATION OF WATER-SOLUBLE O-PHOSPHONOOXYMETHYL PRODRUGS
  IMPROVED PROCESS FOR THE PREPARATION OF WATER-SOLUBLE O-PHOSPHONOOXYMETHYL PRODRUGS