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LT - PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE
EN - PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 413/06
C07D 265/32
European patent
(11) Number of the document 1499611
(13) Kind of document T
(96) European patent application number 03726338.1
Date of filing the European patent application 2003-04-17
(97) Date of publication of the European application 2005-01-26
(45) Date of publication and mention of the grant of the patent 2015-02-11
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2003/011956
Date 2003-04-17
PCT application publication
(87) Number WO 2003/089429
Date 2003-10-30
Priority applications
(30) Number Date Country code
373734 P 2002-04-18 US
Inventors
(72)
HUFFMAN, Mark, US
KABA, Mahmoud, S., US
PAYACK, Joseph, F., US
HANDS, David, GB
Grantee
(73) MERCK SHARP & DOHME LTD., Hertford Road, Hoddesdon, Hertfordshire EN11 9BU, GB
Merck Sharp & Dohme Corp., 126 East Lincoln Avenue, Rahway, NJ 07065-0907, US
Title
(54) PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE
  PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE