LT - PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE
EN - PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 413/06 |
|
|
|
C07D 265/32 |
|
European patent
| (11) |
Number of the document |
1499611 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
03726338.1 |
|
Date of filing the European patent application |
2003-04-17 |
| (97) |
Date of publication of the European application |
2005-01-26 |
| (45) |
Date of publication and mention of the grant of the patent |
2015-02-11
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/US2003/011956 |
|
Date |
2003-04-17 |
PCT application publication
| (87) |
Number |
WO 2003/089429 |
|
Date |
2003-10-30 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
373734 P |
2002-04-18
|
US |
Inventors
| (72) |
HUFFMAN, Mark, US
KABA, Mahmoud, S., US
PAYACK, Joseph, F., US
HANDS, David, GB
|
Grantee
| (73) |
MERCK SHARP & DOHME LTD.,
Hertford Road, Hoddesdon, Hertfordshire EN11 9BU,
GB
Merck Sharp & Dohme Corp.,
126 East Lincoln Avenue, Rahway, NJ 07065-0907,
US
|
Title
| (54) |
PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE |
| |
PROCESS FOR 5-2(R)-1(R)-3,5-BIS(TRIFLUOROMETHYL)PHENYL ETHOXY -3(S)-(4-FLUOROPHENYL)-4-MORPHOLINYL METHYL -1,2-DIHYDRO-3H-1,2,4-TRIAZOL-3-ONE |