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LT - POLYMORPHIC FORMS OF THE PHOSPHATE SALT OF 8-FLUORO-2-{4-[(METHYLAMINO)METHYL]PHENYL}-1,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3-CD]INDOL-6-ONE
EN - POLYMORPHIC FORMS OF THE PHOSPHATE SALT OF 8-FLUORO-2-{4-[(METHYLAMINO)METHYL]PHENYL}-1,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3-CD]INDOL-6-ONE

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 487/06
A61K 31/55
A61P 35/00
A61P 25/00
Europos patentas
(11) Patento numeris 1799685
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 05799991.4
Europos patento paraiškos padavimo data 2005-09-12
(97) Europos patento paraiškos paskelbimo data 2007-06-27
(45) Paskelbimo apie Europos patento išdavimą data 2012-03-28
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/IB2005/002941
Data 2005-09-12
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2006/033007
Data 2006-03-30
Prioriteto paraiškos
(30) Numeris Data Šalis
612459 P 2004-09-22 US
679296 P 2005-05-09 US
Išradėjai
(72)
LIU, Jia, Agouron Pharmaceuticals, Inc., US
NAYYAR, Naresh, Agouron Pharmaceuticals, Inc., US
GUO, Ming Agouron Pharmaceuticals, Inc. A Pfizer Company, US
WU, Zhen-Ping, Agouron Pharmaceuticals, Inc., US
BORER Bennett C., Agouron Pharmaceuticals, Inc., US
SRIRANGAM, A.N., Agouron Pharmaceuticals, Inc., US
MITCHELL, Mark B., Agouron Pharmaceuticals, Inc., US
LI, Yi, Agouron Pharmaceuticals, Inc., US
CHU, Jan-Jon, Agouron Pharmaceuticals, Inc., US
Savininkas
(73) Cancer Research Technology Limited, Sardinia House, Sardinia Street, London WC2A 3NL, GB
Pfizer Inc., 235 East 42nd Street, New York, NY 10017, US
Pavadinimas
(54) POLYMORPHIC FORMS OF THE PHOSPHATE SALT OF 8-FLUORO-2-{4-[(METHYLAMINO)METHYL]PHENYL}-1,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3-CD]INDOL-6-ONE
  POLYMORPHIC FORMS OF THE PHOSPHATE SALT OF 8-FLUORO-2-{4-[(METHYLAMINO)METHYL]PHENYL}-1,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3-CD]INDOL-6-ONE