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LT - PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID
EN - PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61P 29/00
A61K 31/675
C07F 9/6558
European patent
(11) Number of the document 1809379
(13) Kind of document T
(96) European patent application number 05851364.9
Date of filing the European patent application 2005-11-03
(97) Date of publication of the European application 2007-07-25
(45) Date of publication and mention of the grant of the patent 2011-10-19
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2005/039946
Date 2005-11-03
PCT application publication
(87) Number WO 2006/060110
Date 2006-06-08
Priority applications
(30) Number Date Country code
625209 P 2004-11-05 US
Inventors
(72)
MCNAMARA, James, Michael, US
MATTY, Louis, US
ROSEN, Jonathan, D., US
Grantee
(73) Merck Sharp & Dohme Corp., 126 East Lincoln Avenue, Rahway, NJ 07065, US
Title
(54) PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID
  PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID