LT - PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID
EN - PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
A61P 29/00 |
|
|
|
A61K 31/675 |
|
|
|
C07F 9/6558 |
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European patent
| (11) |
Number of the document |
1809379 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
05851364.9 |
|
Date of filing the European patent application |
2005-11-03 |
| (97) |
Date of publication of the European application |
2007-07-25 |
| (45) |
Date of publication and mention of the grant of the patent |
2011-10-19
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/US2005/039946 |
|
Date |
2005-11-03 |
PCT application publication
| (87) |
Number |
WO 2006/060110 |
|
Date |
2006-06-08 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
625209 P |
2004-11-05
|
US |
Inventors
| (72) |
MCNAMARA, James, Michael, US
MATTY, Louis, US
ROSEN, Jonathan, D., US
|
Grantee
| (73) |
Merck Sharp & Dohme Corp.,
126 East Lincoln Avenue, Rahway, NJ 07065,
US
|
Title
| (54) |
PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID |
| |
PROCESS FOR PREPARING (3-(2(R)-((1R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-3(S)-(4-FLUOROPHENYL)MORPHOLIN-4-YL)METHYL)-5-OXO-4,5-DIHYDRO-(1,2,4)-TRIAZOL-1-YL) PHOSPHONIC ACID |