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LT - N-HYDROXY-3-(4-{3-PHENYL-3-OXO-PROPENYL}-PHENYL)-ACRYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF CANCER
EN - N-HYDROXY-3-(4-{3-PHENYL-3-OXO-PROPENYL}-PHENYL)-ACRYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF CANCER

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 295/10
C07D 211/58
C07D 295/18
C07D 295/22
C07D 295/20
C07D 211/46
C07D 213/54
A61K 31/495
A61K 31/4468
A61K 31/5375
A61P 35/00
European patent
(11) Number of the document 2049508
(13) Kind of document T
(96) European patent application number 07727569.1
Date of filing the European patent application 2007-03-30
(97) Date of publication of the European application 2009-04-22
(45) Date of publication and mention of the grant of the patent 2010-06-09
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2007/053097
Date 2007-03-30
PCT application publication
(87) Number WO 2007/113249
Date 2007-10-11
Priority applications
(30) Number Date Country code
MI20060621 2006-03-31 IT
Inventors
(72)
MAI, Antonello, IT
MINUCCI, Saverio, IT
THALER, Florian, IT
PAIN, Gilles, IT
COLOMBO, Andrea, IT
GAGLIARDI, Stefania, IT
Grantee
(73) DAC S.r.l., Piazzetta Maurilio Bossi 4, 20121 Milano, IT
Title
(54) N-HYDROXY-3-(4-{3-PHENYL-3-OXO-PROPENYL}-PHENYL)-ACRYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF CANCER
  N-HYDROXY-3-(4-{3-PHENYL-3-OXO-PROPENYL}-PHENYL)-ACRYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF CANCER