LT - POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR
EN - POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
(51) |
INT.CL. |
C07D 401/04 |
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A61K 31/513 |
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A61P 9/00 |
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European patent
(11) |
Number of the document |
2102185 |
(13) |
Kind of document |
T |
(96) |
European patent application number |
07864915.9 |
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Date of filing the European patent application |
2007-11-29 |
(97) |
Date of publication of the European application |
2009-09-23 |
(45) |
Date of publication and mention of the grant of the patent |
2012-08-15
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(46) |
Date of publication of the claims translation |
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PCT application
(86) |
Number |
PCT/US2007/085933 |
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Date |
2007-11-29 |
PCT application publication
(87) |
Number |
WO 2008/067465 |
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Date |
2008-06-05 |
Priority applications
(30) |
Number |
Date |
Country code |
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867764 P |
2006-11-29
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US |
Inventors
(72) |
KELLY, Ron C., US
KOZTECKI, Lien H., US
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Grantee
(73) |
Takeda Pharmaceutical Company Limited,
1-1, Doshomachi 4-chome Chuo-ku, Osaka- shi, Osaka 541-0045,
JP
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Title
(54) |
POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR |
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POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR |