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LT - POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR
EN - POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 401/04
A61K 31/513
A61P 9/00
European patent
(11) Number of the document 2102185
(13) Kind of document T
(96) European patent application number 07864915.9
Date of filing the European patent application 2007-11-29
(97) Date of publication of the European application 2009-09-23
(45) Date of publication and mention of the grant of the patent 2012-08-15
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2007/085933
Date 2007-11-29
PCT application publication
(87) Number WO 2008/067465
Date 2008-06-05
Priority applications
(30) Number Date Country code
867764 P 2006-11-29 US
Inventors
(72)
KELLY, Ron C., US
KOZTECKI, Lien H., US
Grantee
(73) Takeda Pharmaceutical Company Limited, 1-1, Doshomachi 4-chome Chuo-ku, Osaka- shi, Osaka 541-0045, JP
Title
(54) POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR
  POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR