LT - POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR
EN - POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 401/04 |
|
|
|
A61K 31/513 |
|
|
|
A61P 9/00 |
|
European patent
| (11) |
Number of the document |
2102185 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
07864915.9 |
|
Date of filing the European patent application |
2007-11-29 |
| (97) |
Date of publication of the European application |
2009-09-23 |
| (45) |
Date of publication and mention of the grant of the patent |
2012-08-15
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/US2007/085933 |
|
Date |
2007-11-29 |
PCT application publication
| (87) |
Number |
WO 2008/067465 |
|
Date |
2008-06-05 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
867764 P |
2006-11-29
|
US |
Inventors
| (72) |
KELLY, Ron C., US
KOZTECKI, Lien H., US
|
Grantee
| (73) |
Takeda Pharmaceutical Company Limited,
1-1, Doshomachi 4-chome Chuo-ku, Osaka- shi, Osaka 541-0045,
JP
|
Title
| (54) |
POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR |
| |
POLYMORPHS OF SUCCINATE SALT OF 2-[6-(3-AMINO-PIPERIDIN-1-YL)-3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YLMETHY]-4-FLUOR-BENZONITRILE AND METHODS OF USE THEREFOR |