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LT - NOVEL CRYSTALS AND PROCESS OF MAKING 5-({[2-AMINO-3-(4-CARBAMOYL-2,6-DIMETHYL-PHENYL)-PROPIONYL]-[1-(4-PHENYL-1H-IMIDAZOL-2-YL)-ETHYL]-AMINO}-METHYL)-2-METHOXY- BENZOIC ACID
EN - NOVEL CRYSTALS AND PROCESS OF MAKING 5-({[2-AMINO-3-(4-CARBAMOYL-2,6-DIMETHYL-PHENYL)-PROPIONYL]-[1-(4-PHENYL-1H-IMIDAZOL-2-YL)-ETHYL]-AMINO}-METHYL)-2-METHOXY- BENZOIC ACID

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 233/64
A61K 31/4164
A61P 1/00
European patent
(11) Number of the document 2176234
(13) Kind of document T
(96) European patent application number 08781434.9
Date of filing the European patent application 2008-07-07
(97) Date of publication of the European application 2010-04-21
(45) Date of publication and mention of the grant of the patent 2016-01-27
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2008/069318
Date 2008-07-07
PCT application publication
(87) Number WO 2009/009480
Date 2009-01-15
Priority applications
(30) Number Date Country code
948584 P 2007-07-09 US
Inventors
(72)
ANZALONE, Luigi, US
VILLANI, Frank J., US
TELEHA, Christopher Allan, US
FEIBUSH, Penina, US
FEGELY, Barry, US
Grantee
(73) Forest Tosara Limited, Unit 146 Baldoyle Industrial Estate Grange Road, Baldoyle,Dublin 13, IE
Title
(54) NOVEL CRYSTALS AND PROCESS OF MAKING 5-({[2-AMINO-3-(4-CARBAMOYL-2,6-DIMETHYL-PHENYL)-PROPIONYL]-[1-(4-PHENYL-1H-IMIDAZOL-2-YL)-ETHYL]-AMINO}-METHYL)-2-METHOXY- BENZOIC ACID
  NOVEL CRYSTALS AND PROCESS OF MAKING 5-({[2-AMINO-3-(4-CARBAMOYL-2,6-DIMETHYL-PHENYL)-PROPIONYL]-[1-(4-PHENYL-1H-IMIDAZOL-2-YL)-ETHYL]-AMINO}-METHYL)-2-METHOXY- BENZOIC ACID