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LT - SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE
EN - SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 403/12
A61K 31/506
A61P 1/00
A61P 25/00
European patent
(11) Number of the document 2203444
(13) Kind of document T
(96) European patent application number 08834252.2
Date of filing the European patent application 2008-09-25
(97) Date of publication of the European application 2010-07-07
(45) Date of publication and mention of the grant of the patent 2013-07-24
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2008/077594
Date 2008-09-25
PCT application publication
(87) Number WO 2009/042733
Date 2009-04-02
Priority applications
(30) Number Date Country code
975846 P 2007-09-28 US
Inventors
(72)
BEDNARZ, Mark, S., US
DE PAUL, Susan, CH
KANAMARLAPUDI, Ramanaiah, C., US
PERLBERG, Anett, CH
ZHANG, Haiming, US
Grantee
(73) Lexicon Pharmaceuticals, Inc., 8800 Technology Forest Place, The Woodlands, TX 77381, US
Title
(54) SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE
  SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE