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Legal status
Patent not validated
| (51) | INT.CL. | C07D 403/12 | |
| A61K 31/506 | |||
| A61P 1/00 | |||
| A61P 25/00 |
| (11) | Number of the document | 2203444 |
| (13) | Kind of document | T |
| (96) | European patent application number | 08834252.2 |
| Date of filing the European patent application | 2008-09-25 | |
| (97) | Date of publication of the European application | 2010-07-07 |
| (45) | Date of publication and mention of the grant of the patent | 2013-07-24 |
| (46) | Date of publication of the claims translation |
| (86) | Number | PCT/US2008/077594 |
| Date | 2008-09-25 |
| (87) | Number | WO 2009/042733 |
| Date | 2009-04-02 |
| (30) | Number | Date | Country code |
| 975846 P | 2007-09-28 | US |
| (72) |
BEDNARZ, Mark, S., US
DE PAUL, Susan, CH
KANAMARLAPUDI, Ramanaiah, C., US
PERLBERG, Anett, CH
ZHANG, Haiming, US
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| (73) |
Lexicon Pharmaceuticals, Inc.,
8800 Technology Forest Place, The Woodlands, TX 77381,
US
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| (54) | SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE |
| SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE |