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Legal status
Patent not validated
(51) | INT.CL. | C07D 403/12 | |
A61K 31/506 | |||
A61P 1/00 | |||
A61P 25/00 |
(11) | Number of the document | 2203444 |
(13) | Kind of document | T |
(96) | European patent application number | 08834252.2 |
Date of filing the European patent application | 2008-09-25 | |
(97) | Date of publication of the European application | 2010-07-07 |
(45) | Date of publication and mention of the grant of the patent | 2013-07-24 |
(46) | Date of publication of the claims translation |
(86) | Number | PCT/US2008/077594 |
Date | 2008-09-25 |
(87) | Number | WO 2009/042733 |
Date | 2009-04-02 |
(30) | Number | Date | Country code |
975846 P | 2007-09-28 | US |
(72) |
BEDNARZ, Mark, S., US
DE PAUL, Susan, CH
KANAMARLAPUDI, Ramanaiah, C., US
PERLBERG, Anett, CH
ZHANG, Haiming, US
|
(73) |
Lexicon Pharmaceuticals, Inc.,
8800 Technology Forest Place, The Woodlands, TX 77381,
US
|
(54) | SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE |
SOLIDS FORMS OF ( S) -ETHYL 2-AMIN0-3- (4- (2 -AMINO- 6- ( (R) -1- (4-CHL0R0-2- O-METHYL-IH-PYRAZOL- 1-YL) PHENYL) -2, 2, 2-TRIFLUORETHOXY) -PYRIMIDIN-4-YL) PHENYL) PROPANOATE |