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LT - (+)-1,4-DIHYDRO-7-[(3S,4S)-3-METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID IN COMBINATION WITH GEMCITABINE FOR USE IN TREATING CANCER
EN - (+)-1,4-DIHYDRO-7-[(3S,4S)-3-METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID IN COMBINATION WITH GEMCITABINE FOR USE IN TREATING CANCER

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/282
A61K 31/4178
A61K 31/4375
A61K 31/555
A61P 35/00
European patent
(11) Number of the document 2214662
(13) Kind of document T
(96) European patent application number 08843165.5
Date of filing the European patent application 2008-10-21
(97) Date of publication of the European application 2010-08-11
(45) Date of publication and mention of the grant of the patent 2016-07-13
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2008/011960
Date 2008-10-21
PCT application publication
(87) Number WO 2009/054935
Date 2009-04-30
Priority applications
(30) Number Date Country code
981766 P 2007-10-22 US
Inventors
(72)
SILVERMAN, Jeffrey, A., US
Grantee
(73) Sunesis Pharmaceuticals, Inc., 395 Oyster Point Blvd., South San Francisco, CA 94080, US
Title
(54) (+)-1,4-DIHYDRO-7-[(3S,4S)-3-METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID IN COMBINATION WITH GEMCITABINE FOR USE IN TREATING CANCER
  (+)-1,4-DIHYDRO-7-[(3S,4S)-3-METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID IN COMBINATION WITH GEMCITABINE FOR USE IN TREATING CANCER