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LT - CRYSTALLINE FORMS AND TWO SOLVATED FORMS OF 4-AMINO-5-FLUORO-3-[5-(4-METHYLPIPERAZIN-1-YL)-1H-BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE LACTIC ACID SALTS
EN - CRYSTALLINE FORMS AND TWO SOLVATED FORMS OF 4-AMINO-5-FLUORO-3-[5-(4-METHYLPIPERAZIN-1-YL)-1H-BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE LACTIC ACID SALTS

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 401/14
A61K 31/496
A61P 35/00
European patent
(11) Number of the document 2257544
(13) Kind of document T
(96) European patent application number 09721534.7
Date of filing the European patent application 2009-03-18
(97) Date of publication of the European application 2010-12-08
(45) Date of publication and mention of the grant of the patent 2014-12-03
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2009/053222
Date 2009-03-18
PCT application publication
(87) Number WO 2009/115562
Date 2009-09-24
Priority applications
(30) Number Date Country code
37746 P 2008-03-19 US
Inventors
(72)
GIRON, Danielle, FR
HAMMERSCHMIDT, Walter, CH
PIECHON, Philippe, FR
POLASEK, Johanne, CH
SCHREINER, Andreas, CH
STOWASSER, Frank, DE
Grantee
(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
Title
(54) CRYSTALLINE FORMS AND TWO SOLVATED FORMS OF 4-AMINO-5-FLUORO-3-[5-(4-METHYLPIPERAZIN-1-YL)-1H-BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE LACTIC ACID SALTS
  CRYSTALLINE FORMS AND TWO SOLVATED FORMS OF 4-AMINO-5-FLUORO-3-[5-(4-METHYLPIPERAZIN-1-YL)-1H-BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE LACTIC ACID SALTS