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EN | LT
LT - IMPROVED PROCESS FOR PREPARATION OF (2R)-4-OXO-4-[3- (TRIFLUOROMETHYL)-5,6-DIHYDRO [1,2,4]-TRIAZOLO[4,3-A]PYRAZIN- 7(8H)-YL]-L-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE&NEW IMPURITIES IN PREPARATION THEREOF
EN - IMPROVED PROCESS FOR PREPARATION OF (2R)-4-OXO-4-[3- (TRIFLUOROMETHYL)-5,6-DIHYDRO [1,2,4]-TRIAZOLO[4,3-A]PYRAZIN- 7(8H)-YL]-L-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE&NEW IMPURITIES IN PREPARATION THEREOF

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 487/04
Europos patentas
(11) Patento numeris 2331545
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 09765169.9
Europos patento paraiškos padavimo data 2009-08-26
(97) Europos patento paraiškos paskelbimo data 2011-06-15
(45) Paskelbimo apie Europos patento išdavimą data 2013-10-02
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/IN2009/000470
Data 2009-08-26
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2010/032264
Data 2010-03-25
Prioriteto paraiškos
(30) Numeris Data Šalis
MU17982008 2008-08-27 IN
MU01882009 2009-02-02 IN
MU07852009 2009-03-30 IN
Išradėjai
(72)
KOTHARI, Himanshu, Madhusudan, IN
DAVE, Mayank, Ghanshyambhai, IN
PANDEY, Bipin, IN
SHUKLA, Bhavin, Shriprasad, IN
Savininkas
(73) Cadila Healthcare Limited, Zydus Tower Satellite Cross Roads, Ahmedabad 380 015 Gujarat, IN
Pavadinimas
(54) IMPROVED PROCESS FOR PREPARATION OF (2R)-4-OXO-4-[3- (TRIFLUOROMETHYL)-5,6-DIHYDRO [1,2,4]-TRIAZOLO[4,3-A]PYRAZIN- 7(8H)-YL]-L-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE&NEW IMPURITIES IN PREPARATION THEREOF
  IMPROVED PROCESS FOR PREPARATION OF (2R)-4-OXO-4-[3- (TRIFLUOROMETHYL)-5,6-DIHYDRO [1,2,4]-TRIAZOLO[4,3-A]PYRAZIN- 7(8H)-YL]-L-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE&NEW IMPURITIES IN PREPARATION THEREOF