LT - A PROCESS FOR PREPARING [1S- ]1-ALPHA, 2-ALPHA, 3-BETA (1S*, 2R*) 5-BETA] ]-3- [7- [2- (3, 4-DIF LUOROPHENYL) -CYCLOPROPYLAMINO]- 5- (PROPYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D]PYRIMIDIN-3-YL]-5- (2- HYDROXYETHOXY) CYCLOPENTANE-1, 2-DIOL AND TO ITS INTERM
EN - A PROCESS FOR PREPARING [1S- ]1-ALPHA, 2-ALPHA, 3-BETA (1S*, 2R*) 5-BETA] ]-3- [7- [2- (3, 4-DIF LUOROPHENYL) -CYCLOPROPYLAMINO]- 5- (PROPYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D]PYRIMIDIN-3-YL]-5- (2- HYDROXYETHOXY) CYCLOPENTANE-1, 2-DIOL AND TO ITS INTERM
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 487/04 |
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|
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C07D 317/44 |
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C07D 405/04 |
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C07D 405/12 |
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European patent
| (11) |
Number of the document |
2340252 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
09813307.7 |
|
Date of filing the European patent application |
2009-09-08 |
| (97) |
Date of publication of the European application |
2011-07-06 |
| (45) |
Date of publication and mention of the grant of the patent |
2015-11-11
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/SE2009/050999 |
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Date |
2009-09-08 |
PCT application publication
| (87) |
Number |
WO 2010/030224 |
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Date |
2010-03-18 |
Priority applications
| (30) |
Number |
Date |
Country code |
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95341 P |
2008-09-09
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US |
Inventors
| (72) |
AUFDENBLATTEN, Rhony, CH
BOHLIN, Martin, Hans, GB
HELLSTRÖM, Helena, GB
JOHANSSON, Peter, W, GB
LARSSON, Ulf, G, GB
RECKNAGEL, Mikaela, SE
WEISS, Ursula, heiress of WEISS Andreas (Deceased), CH
|
Grantee
| (73) |
AstraZeneca AB,
151 85 Södertälje,
SE
|
Title
| (54) |
A PROCESS FOR PREPARING [1S- ]1-ALPHA, 2-ALPHA, 3-BETA (1S*, 2R*) 5-BETA] ]-3- [7- [2- (3, 4-DIF LUOROPHENYL) -CYCLOPROPYLAMINO]- 5- (PROPYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D]PYRIMIDIN-3-YL]-5- (2- HYDROXYETHOXY) CYCLOPENTANE-1, 2-DIOL AND TO ITS INTERM |
| |
A PROCESS FOR PREPARING [1S- ]1-ALPHA, 2-ALPHA, 3-BETA (1S*, 2R*) 5-BETA] ]-3- [7- [2- (3, 4-DIF LUOROPHENYL) -CYCLOPROPYLAMINO]- 5- (PROPYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D]PYRIMIDIN-3-YL]-5- (2- HYDROXYETHOXY) CYCLOPENTANE-1, 2-DIOL AND TO ITS INTERM |
