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LT - PROCESS FOR THE PREPARATION OF (3R,3AS,6AR)-HEXAHYDROFURO [2,3-B]FURAN-3-YL (1S,2R)-3-[[(4-AMINOPHENYL) SULFONYL](ISOBUTYL) AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE
EN - PROCESS FOR THE PREPARATION OF (3R,3AS,6AR)-HEXAHYDROFURO [2,3-B]FURAN-3-YL (1S,2R)-3-[[(4-AMINOPHENYL) SULFONYL](ISOBUTYL) AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 493/04
European patent
(11) Number of the document 2346877
(13) Kind of document T
(96) European patent application number 09782438.7
Date of filing the European patent application 2009-09-01
(97) Date of publication of the European application 2011-07-27
(45) Date of publication and mention of the grant of the patent 2014-08-20
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2009/061253
Date 2009-09-01
PCT application publication
(87) Number WO 2010/023322
Date 2010-03-04
Priority applications
(30) Number Date Country code
08163383 2008-09-01 EP
Inventors
(72)
WIGERINCK, Piet Tom Bert Paul, BE
SURLERAUX, Dominique Louis Nestor Ghislain, BE
VERSCHUEREN, Wim Gaston, BE
DE KOCK, Herman Augustinus, BE
AELTERMAN, Wim Albert Alex, BE
Grantee
(73) Janssen R&D Ireland, Eastgate Village, Eastgate, Little Island, County Cork, IE
Title
(54) PROCESS FOR THE PREPARATION OF (3R,3AS,6AR)-HEXAHYDROFURO [2,3-B]FURAN-3-YL (1S,2R)-3-[[(4-AMINOPHENYL) SULFONYL](ISOBUTYL) AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE
  PROCESS FOR THE PREPARATION OF (3R,3AS,6AR)-HEXAHYDROFURO [2,3-B]FURAN-3-YL (1S,2R)-3-[[(4-AMINOPHENYL) SULFONYL](ISOBUTYL) AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE