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LT - N4-(2,2-dimetil-4-[(divandenilio fosfonoksi)metil] -3-okso-5-pirido[1,4]oksazin-6-il)-5-fluor-N2-(3,4,5-trimetoksifenil)-2,4-pirimidindiamino dinatrio druskos sintezė
EN - SYNTHESIS OF N4-(2,2-DIMETHYL-4-[(DIHYDROGEN PHOSPHONOXY)METHYL]-3-OXO-5-PYRIDO[1,4]OXAZIN-6-YL)-5-FLUORO-N2-(3,4,5-TRIMETHOXYPHENYL)-2,4-PYRIMIDINEDIAMINE DISODIUM SALT

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Patent in force

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07F 9/6561 (2006.01)
European patent
(11) Number of the document 2448950
(13) Kind of document T
(96) European patent application number 10730679.7
Date of filing the European patent application 2010-07-01
(97) Date of publication of the European application 2012-05-09
(45) Date of publication and mention of the grant of the patent 2016-01-13
(46) Date of publication of the claims translation 2016-04-11
PCT application
(86) Number PCT/US2010/040792
Date 2010-07-01
PCT application publication
(87) Number WO 2011/002999
Date 2011-01-06
Priority applications
(30) Number Date Country code
270073 P 2009-07-02 US
Inventors
(72)
FELFER, Ulfried, AT
GISELBRECHT, Karl-Heinz, AT
WOLBERG, Michael, DE
Grantee
(73) Rigel Pharmaceuticals, Inc., 1180 Veterans Boulevard, South San Francisco, CA 94080, US
Attorney or representative
(74) Liudmila GERASIMOVIČ, IĮ "Liudmila Gerasimovič, Patentinis patikėtinis", Vingrių g. 13-42, LT-01141 Vilnius, LT
Title
(54) N4-(2,2-dimetil-4-[(divandenilio fosfonoksi)metil] -3-okso-5-pirido[1,4]oksazin-6-il)-5-fluor-N2-(3,4,5-trimetoksifenil)-2,4-pirimidindiamino dinatrio druskos sintezė
  SYNTHESIS OF N4-(2,2-DIMETHYL-4-[(DIHYDROGEN PHOSPHONOXY)METHYL]-3-OXO-5-PYRIDO[1,4]OXAZIN-6-YL)-5-FLUORO-N2-(3,4,5-TRIMETHOXYPHENYL)-2,4-PYRIMIDINEDIAMINE DISODIUM SALT
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2025-06-18 16 347.00 EUR
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2026-07-01