LT - N4-(2,2-dimetil-4-[(divandenilio fosfonoksi)metil] -3-okso-5-pirido[1,4]oksazin-6-il)-5-fluor-N2-(3,4,5-trimetoksifenil)-2,4-pirimidindiamino dinatrio druskos sintezė
EN - SYNTHESIS OF N4-(2,2-DIMETHYL-4-[(DIHYDROGEN PHOSPHONOXY)METHYL]-3-OXO-5-PYRIDO[1,4]OXAZIN-6-YL)-5-FLUORO-N2-(3,4,5-TRIMETHOXYPHENYL)-2,4-PYRIMIDINEDIAMINE DISODIUM SALT
Legal status
Patent in force
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07F 9/6561 |
(2006.01) |
European patent
| (11) |
Number of the document |
2448950 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
10730679.7 |
|
Date of filing the European patent application |
2010-07-01 |
| (97) |
Date of publication of the European application |
2012-05-09 |
| (45) |
Date of publication and mention of the grant of the patent |
2016-01-13
|
| (46) |
Date of publication of the claims translation |
2016-04-11
|
PCT application
| (86) |
Number |
PCT/US2010/040792 |
|
Date |
2010-07-01 |
PCT application publication
| (87) |
Number |
WO 2011/002999 |
|
Date |
2011-01-06 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
270073 P |
2009-07-02
|
US |
Inventors
| (72) |
FELFER, Ulfried, AT
GISELBRECHT, Karl-Heinz, AT
WOLBERG, Michael, DE
|
Grantee
| (73) |
Rigel Pharmaceuticals, Inc.,
1180 Veterans Boulevard, South San Francisco, CA 94080,
US
|
Attorney or representative
| (74) |
Liudmila GERASIMOVIČ,
IĮ "Liudmila Gerasimovič, Patentinis patikėtinis", Vingrių g. 13-42, LT-01141 Vilnius,
LT
|
Title
| (54) |
N4-(2,2-dimetil-4-[(divandenilio fosfonoksi)metil] -3-okso-5-pirido[1,4]oksazin-6-il)-5-fluor-N2-(3,4,5-trimetoksifenil)-2,4-pirimidindiamino dinatrio druskos sintezė |
| |
SYNTHESIS OF N4-(2,2-DIMETHYL-4-[(DIHYDROGEN PHOSPHONOXY)METHYL]-3-OXO-5-PYRIDO[1,4]OXAZIN-6-YL)-5-FLUORO-N2-(3,4,5-TRIMETHOXYPHENYL)-2,4-PYRIMIDINEDIAMINE DISODIUM SALT |
Last renewal fee
|
Payment date |
Validity (years) |
Amount |
|
2025-06-18 |
16 |
347.00
EUR
|
Next renewal fee
|
2026-07-01 |