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LT - PROCESS FOR PRODUCING CRYSTALS OF POLYMORPHIC 2-(3-CYANO-4-ISOBUTYLOXYPHENYL)-4-METHYL-5-THIAZOLECARBOXYLIC ACID BY POOR-SOLVENT ADDITION METHOD
EN - PROCESS FOR PRODUCING CRYSTALS OF POLYMORPHIC 2-(3-CYANO-4-ISOBUTYLOXYPHENYL)-4-METHYL-5-THIAZOLECARBOXYLIC ACID BY POOR-SOLVENT ADDITION METHOD

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 277/20
A61K 31/426
A61P 19/06
C07D 277/56
European patent
(11) Number of the document 2455372
(13) Kind of document T
(96) European patent application number 10799952.6
Date of filing the European patent application 2010-07-14
(97) Date of publication of the European application 2012-05-23
(45) Date of publication and mention of the grant of the patent 2017-10-11
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/JP2010/062291
Date 2010-07-14
PCT application publication
(87) Number WO 2011/007895
Date 2011-01-20
Priority applications
(30) Number Date Country code
2009166755 2009-07-15 JP
Inventors
(72)
UEMURA, Akihito, JP
NOGATA, Tomoaki, JP
TAKEYASU, Takumi, JP
Grantee
(73) Teijin Pharma Limited, 2-1, Kasumigaseki 3-chome Chiyoda-ku, Tokyo 100-0013, JP
Title
(54) PROCESS FOR PRODUCING CRYSTALS OF POLYMORPHIC 2-(3-CYANO-4-ISOBUTYLOXYPHENYL)-4-METHYL-5-THIAZOLECARBOXYLIC ACID BY POOR-SOLVENT ADDITION METHOD
  PROCESS FOR PRODUCING CRYSTALS OF POLYMORPHIC 2-(3-CYANO-4-ISOBUTYLOXYPHENYL)-4-METHYL-5-THIAZOLECARBOXYLIC ACID BY POOR-SOLVENT ADDITION METHOD