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LT - OXAZINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS
EN - OXAZINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 265/30
C07D 413/12
C07D 417/12
C07D 471/04
C07D 487/04
A61K 31/5377
A61K 31/553
A61P 25/00
A61P 9/00
European patent
(11) Number of the document 2456763
(13) Kind of document T
(96) European patent application number 10737870.5
Date of filing the European patent application 2010-07-23
(97) Date of publication of the European application 2012-05-30
(45) Date of publication and mention of the grant of the patent 2015-01-21
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2010/060718
Date 2010-07-23
PCT application publication
(87) Number WO 2011/009943
Date 2011-01-27
Priority applications
(30) Number Date Country code
228472 P 2009-07-24 US
258911 P 2009-11-06 US
363702 P 2010-07-13 US
Inventors
(72)
BADIGER, Sangamesh, IN
CHEBROLU, Murali, IN
FREDERIKSEN, Mathias, CH
HOLZER, Philipp, CH
HURTH, Konstanze, CH
LUEOEND, Rainer Martin, CH
MACHAUER, Rainer, CH
MOEBITZ, Henrik, CH
NEUMANN, Ulf, CH
RAMOS, Rita, CH
RUEEGER, Heinrich, CH
TINTELNOT-BLOMLEY, Marina, CH
VEENSTRA, Siem Jacob, CH
VOEGTLE, Markus, CH
SCHAEFER, Michael, CH
Grantee
(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
Title
(54) OXAZINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS
  OXAZINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS