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Legal status
Patent not validated
| (51) | INT.CL. | C07D 265/30 | |
| C07D 413/12 | |||
| C07D 417/12 | |||
| C07D 471/04 | |||
| C07D 487/04 | |||
| A61K 31/5377 | |||
| A61K 31/553 | |||
| A61P 25/00 | |||
| A61P 9/00 |
| (11) | Number of the document | 2456763 |
| (13) | Kind of document | T |
| (96) | European patent application number | 10737870.5 |
| Date of filing the European patent application | 2010-07-23 | |
| (97) | Date of publication of the European application | 2012-05-30 |
| (45) | Date of publication and mention of the grant of the patent | 2015-01-21 |
| (46) | Date of publication of the claims translation |
| (86) | Number | PCT/EP2010/060718 |
| Date | 2010-07-23 |
| (87) | Number | WO 2011/009943 |
| Date | 2011-01-27 |
| (30) | Number | Date | Country code |
| 228472 P | 2009-07-24 | US | |
| 258911 P | 2009-11-06 | US | |
| 363702 P | 2010-07-13 | US |
| (72) |
BADIGER, Sangamesh, IN
CHEBROLU, Murali, IN
FREDERIKSEN, Mathias, CH
HOLZER, Philipp, CH
HURTH, Konstanze, CH
LUEOEND, Rainer Martin, CH
MACHAUER, Rainer, CH
MOEBITZ, Henrik, CH
NEUMANN, Ulf, CH
RAMOS, Rita, CH
RUEEGER, Heinrich, CH
TINTELNOT-BLOMLEY, Marina, CH
VEENSTRA, Siem Jacob, CH
VOEGTLE, Markus, CH
SCHAEFER, Michael, CH
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| (73) |
Novartis AG,
Lichtstrasse 35, 4056 Basel,
CH
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| (54) | OXAZINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS |
| OXAZINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS |