LT - Process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4 H-imidazo[1,2-a][1,4]benzodiazepine-4-yl] propionic acid methyl ester or the benzene sulfonate salt thereof, and compounds useful in that process
EN - Process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4 H-imidazo[1,2-a][1,4]benzodiazepine-4-yl] propionic acid methyl ester or the benzene sulfonate salt thereof, and compounds useful in that process
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
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INT.CL. |
C07D 213/16 |
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C07D 213/18 |
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C07D 401/04 |
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C07D 487/04 |
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Europos patentas
| (11) |
Patento numeris |
2477967 |
| (13) |
Dokumento rūšis |
T |
| (96) |
Europos patento paraiškos numeris |
10760917.4 |
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Europos patento paraiškos padavimo data |
2010-09-15 |
| (97) |
Europos patento paraiškos paskelbimo data |
2012-07-25 |
| (45) |
Paskelbimo apie Europos patento išdavimą data |
2015-11-11
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Apibrėžties vertimo paskelbimo data |
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Tarptautinės paraiškos padavimo
| (86) |
Numeris |
PCT/EP2010/005668 |
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Data |
2010-09-15 |
Tarptautinės paraiškos paskelbimo
| (87) |
Numeris |
WO 2011/032692 |
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Data |
2011-03-24 |
Prioriteto paraiškos
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Numeris |
Data |
Šalis |
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09011914 |
2009-09-18
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EP |
Išradėjai
| (72) |
TILBROOK, Stuart, Gary, GB
SCHUMACHER, Andreas, DE
EMMENEGGER, René, CH
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Savininkas
| (73) |
PAION UK Limited,
Compass House Vision Park Chivers way, Cambridge Cambridgeshire CB4 9ZR,
GB
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Pavadinimas
| (54) |
Process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4 H-imidazo[1,2-a][1,4]benzodiazepine-4-yl] propionic acid methyl ester or the benzene sulfonate salt thereof, and compounds useful in that process |
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Process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4 H-imidazo[1,2-a][1,4]benzodiazepine-4-yl] propionic acid methyl ester or the benzene sulfonate salt thereof, and compounds useful in that process |