LT - PROCESS FOR PREPARATION OF 3-(2-HYDROXY-5-SUBSTITUTED PHENYL)-3-PHENYLPROPYLAMINES, INTERMEDIATES FOR MAKING HYDROXYTOLTERODINE AND FESOTERODINE
EN - PROCESS FOR PREPARATION OF 3-(2-HYDROXY-5-SUBSTITUTED PHENYL)-3-PHENYLPROPYLAMINES, INTERMEDIATES FOR MAKING HYDROXYTOLTERODINE AND FESOTERODINE
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07C 45/48 |
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C07C 213/08 |
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C07C 227/16 |
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C07C 47/565 |
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C07C 215/54 |
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C07C 229/36 |
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C07C 219/28 |
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C07C 221/00 |
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C07C 51/41 |
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European patent
| (11) |
Number of the document |
2545024 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
11709079.5 |
|
Date of filing the European patent application |
2011-03-08 |
| (97) |
Date of publication of the European application |
2013-01-16 |
| (45) |
Date of publication and mention of the grant of the patent |
2016-08-03
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| (46) |
Date of publication of the claims translation |
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PCT application
| (86) |
Number |
PCT/EP2011/053465 |
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Date |
2011-03-08 |
PCT application publication
| (87) |
Number |
WO 2011/110556 |
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Date |
2011-09-15 |
Priority applications
| (30) |
Number |
Date |
Country code |
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10155864 |
2010-03-09
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EP |
Inventors
| (72) |
STERK, Damjan, SI
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Grantee
| (73) |
LEK Pharmaceuticals d.d.,
Verovskova 57, 1526 Ljubljana,
SI
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Title
| (54) |
PROCESS FOR PREPARATION OF 3-(2-HYDROXY-5-SUBSTITUTED PHENYL)-3-PHENYLPROPYLAMINES, INTERMEDIATES FOR MAKING HYDROXYTOLTERODINE AND FESOTERODINE |
| |
PROCESS FOR PREPARATION OF 3-(2-HYDROXY-5-SUBSTITUTED PHENYL)-3-PHENYLPROPYLAMINES, INTERMEDIATES FOR MAKING HYDROXYTOLTERODINE AND FESOTERODINE |