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LT - (3-METHYLPYRROLIDIN-3-YL)METHYL PYRIDINYL ETHER DERIVATIVES AND THEIR USE AS NK-3 RECEPTOR ANTAGONISTS
EN - (3-METHYLPYRROLIDIN-3-YL)METHYL PYRIDINYL ETHER DERIVATIVES AND THEIR USE AS NK-3 RECEPTOR ANTAGONISTS

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 401/12
C07D 401/14
C07D 405/14
C07D 413/14
A61K 31/4439
A61P 25/00
European patent
(11) Number of the document 2590963
(13) Kind of document T
(96) European patent application number 11728862.1
Date of filing the European patent application 2011-07-04
(97) Date of publication of the European application 2013-05-15
(45) Date of publication and mention of the grant of the patent 2014-12-03
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2011/061168
Date 2011-07-04
PCT application publication
(87) Number WO 2012/004207
Date 2012-01-12
Priority applications
(30) Number Date Country code
10168688 2010-07-07 EP
Inventors
(72)
NETTEKOVEN, Matthias, DE
RATNI, Hasane, FR
VIFIAN, Walter, CH
Grantee
(73) F. Hoffmann-La Roche AG, Grenzacherstrasse 124, 4070 Basel, CH
Title
(54) (3-METHYLPYRROLIDIN-3-YL)METHYL PYRIDINYL ETHER DERIVATIVES AND THEIR USE AS NK-3 RECEPTOR ANTAGONISTS
  (3-METHYLPYRROLIDIN-3-YL)METHYL PYRIDINYL ETHER DERIVATIVES AND THEIR USE AS NK-3 RECEPTOR ANTAGONISTS