LT - CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT
EN - CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 471/06 |
|
|
|
A61K 31/5025 |
|
|
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A61P 35/00 |
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European patent
| (11) |
Number of the document |
2630146 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
11777005.7 |
|
Date of filing the European patent application |
2011-10-20 |
| (97) |
Date of publication of the European application |
2013-08-28 |
| (45) |
Date of publication and mention of the grant of the patent |
2020-07-01
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/US2011/057039 |
|
Date |
2011-10-20 |
PCT application publication
| (87) |
Number |
WO 2012/054698 |
|
Date |
2012-04-26 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
405476 P |
2010-10-21
|
US |
Inventors
| (72) |
WANG, Bing, US
CHU, Daniel, US
LIU, Yongbo, CN
PENG, Shichun, CN
|
Grantee
| (73) |
Medivation Technologies LLC,
525 Market St., 28th Floor, San Francisco, CA 94105,
US
|
Title
| (54) |
CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT |
| |
CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT |