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LT - CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT
EN - CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 471/06
A61K 31/5025
A61P 35/00
European patent
(11) Number of the document 2630146
(13) Kind of document T
(96) European patent application number 11777005.7
Date of filing the European patent application 2011-10-20
(97) Date of publication of the European application 2013-08-28
(45) Date of publication and mention of the grant of the patent 2020-07-01
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2011/057039
Date 2011-10-20
PCT application publication
(87) Number WO 2012/054698
Date 2012-04-26
Priority applications
(30) Number Date Country code
405476 P 2010-10-21 US
Inventors
(72)
WANG, Bing, US
CHU, Daniel, US
LIU, Yongbo, CN
PENG, Shichun, CN
Grantee
(73) Medivation Technologies LLC, 525 Market St., 28th Floor, San Francisco, CA 94105, US
Title
(54) CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT
  CRYSTALINE (8S,9R)-5-FLUORO-8-(4-FLUOROPHENYL)-9-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-8,9-DIHYDRO-2H-PYRIDO[4,3,2-DE]PHTALAZIN-3(7H)-ONE TOSYLATE SALT