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LT - 5-Chlor-N2-(2-izopropoksi-5-metil-4-piperidin-4-il-fenil)-N4[2-(propan-2-sulfonil)-fenil]-pirimidin-2,4-diamino kristalinės formos
EN - CRYSTALLINE FORMS OF 5-CHLORO-N2-(2-ISOPROPOXY-5-METHYL-4-PIPERIDIN-4-YL-PHENYL)-N4[2-(PROPANE-2-SULFONYL)-PHENYL]-PYRIMIDINE-2,4-DIAMINE

Legal status

Patent revoked (after opposition at EPO)

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 401/12 (2006.01)
A61K 31/506 (2006.01)
A61P 35/00 (2006.01)
European patent
(11) Number of the document 2651918
(13) Kind of document T
(96) European patent application number 11806079.7
Date of filing the European patent application 2011-12-15
(97) Date of publication of the European application 2013-10-23
(45) Date of publication and mention of the grant of the patent 2017-07-12
(46) Date of publication of the claims translation 2017-10-10
PCT application
(86) Number PCT/US2011/065030
Date 2011-12-15
PCT application publication
(87) Number WO 2012/082972
Date 2012-06-21
Priority applications
(30) Number Date Country code
201061424194 P 2010-12-17 US
Inventors
(72)
FENG, Lili, US
GONG, Baoqing, US
KARPINSKI, Piotr H., US
WAYKOLE, Liladhar Murlidhar, US
Grantee
(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
Attorney or representative
(74) Jurga PETNIŪNAITĖ, AAA Law, A. Goštauto g. 40B, Verslo centras "Dvyniai", LT-03163 Vilnius, LT
Title
(54) 5-Chlor-N2-(2-izopropoksi-5-metil-4-piperidin-4-il-fenil)-N4[2-(propan-2-sulfonil)-fenil]-pirimidin-2,4-diamino kristalinės formos
  CRYSTALLINE FORMS OF 5-CHLORO-N2-(2-ISOPROPOXY-5-METHYL-4-PIPERIDIN-4-YL-PHENYL)-N4[2-(PROPANE-2-SULFONYL)-PHENYL]-PYRIMIDINE-2,4-DIAMINE
Last renewal fee
Payment date Validity (years) Amount
2021-11-29 11 289.00 EUR
Legal status
Patent revoked (after opposition at EPO)
Invalidation date 2022-06-01