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LT - SUBSTITUTED METHYLFORMYL REAGENTS AND METHOD OF USING SAME TO MODIFY PHYSICOCHEMICAL AND/OR PHARMACOKINETIC PROPERTIES OF COMPOUNDS
EN - SUBSTITUTED METHYLFORMYL REAGENTS AND METHOD OF USING SAME TO MODIFY PHYSICOCHEMICAL AND/OR PHARMACOKINETIC PROPERTIES OF COMPOUNDS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/11
C07D 401/14
C07D 405/14
C07D 213/80
C07D 213/81
C07D 213/82
C07D 213/803
C07D 401/12
C07D 401/04
C07D 405/12
C07D 471/04
C07D 487/04
C07D 487/22
C07D 491/22
C07D 491/147
C07D 495/14
C07D 295/20
C07D 305/14
European patent
(11) Number of the document 2693876
(13) Kind of document T
(96) European patent application number 12768375.3
Date of filing the European patent application 2012-04-09
(97) Date of publication of the European application 2014-02-12
(45) Date of publication and mention of the grant of the patent 2020-01-15
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/IN2012/000248
Date 2012-04-09
PCT application publication
(87) Number WO 2012/137225
Date 2012-10-11
Priority applications
(30) Number Date Country code
1024DE2011 2011-04-08 IN
Inventors
(72)
DUGAR, Sundeep, US
MAHAJAN, Dinesh, IN
HOLLINGER, Frank, Peter, US
Grantee
(73) Sphaera Pharma Pte. Ltd, 31 Cantonment Road, 089747, Singapore, SG
Title
(54) SUBSTITUTED METHYLFORMYL REAGENTS AND METHOD OF USING SAME TO MODIFY PHYSICOCHEMICAL AND/OR PHARMACOKINETIC PROPERTIES OF COMPOUNDS
  SUBSTITUTED METHYLFORMYL REAGENTS AND METHOD OF USING SAME TO MODIFY PHYSICOCHEMICAL AND/OR PHARMACOKINETIC PROPERTIES OF COMPOUNDS