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LT - Kristalinės (4S,4aS,5aR,12aS)-4-dimetilamino-3,10,12,12a-tetrahidroksi-7-[(metoksi(metil)amino)-metil]-1,11-diokso-1,4,4a,5,5a,6,11,12a-oktahidro-naftacen-2-karboksirūgšties amido druskos ir jų panaudojimo būdai
EN - CRYSTALLINE SALTS OF (4S,4AS,5AR,12AS)-4-DIMETHYLAMINO-3,10,12,12A-TETRAHYDROXY-7-[(METHOXY(METHYL)AMINO)-METHYL]-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDRO-NAPHTHACENE-2-CARBOXYLIC ACID AMIDE AND METHODS OF USING THE SAME

Legal status

Patent lapsed (non-payment of fees)

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/65 (2006.01)
C07C 237/26 (2006.01)
European patent
(11) Number of the document 2707003
(13) Kind of document T
(96) European patent application number 12782600.6
Date of filing the European patent application 2012-05-14
(97) Date of publication of the European application 2014-03-19
(45) Date of publication and mention of the grant of the patent 2019-05-01
(46) Date of publication of the claims translation 2019-10-10
PCT application
(86) Number PCT/US2012/037838
Date 2012-05-14
PCT application publication
(87) Number WO 2012/155146
Date 2012-11-15
Priority applications
(30) Number Date Country code
201161485179 P 2011-05-12 US
Inventors
(72)
COULTER, Catherine, IE
JOHNSTON, Sean, M., US
SEYEDI, Farzaneh, US
Grantee
(73) Allergan Pharmaceuticals International Limited, Clonshaugh Industrial Estate Coolock, Dublin 17, IE
Paratek Pharmaceuticals, Inc., 75 Park Plaza, Boston, MA 02116, US
Attorney or representative
(74) Jurga PETNIŪNAITĖ, AAA Law, A. Goštauto g. 40B, Verslo centras "Dvyniai", LT-03163 Vilnius, LT
Title
(54) Kristalinės (4S,4aS,5aR,12aS)-4-dimetilamino-3,10,12,12a-tetrahidroksi-7-[(metoksi(metil)amino)-metil]-1,11-diokso-1,4,4a,5,5a,6,11,12a-oktahidro-naftacen-2-karboksirūgšties amido druskos ir jų panaudojimo būdai
  CRYSTALLINE SALTS OF (4S,4AS,5AR,12AS)-4-DIMETHYLAMINO-3,10,12,12A-TETRAHYDROXY-7-[(METHOXY(METHYL)AMINO)-METHYL]-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDRO-NAPHTHACENE-2-CARBOXYLIC ACID AMIDE AND METHODS OF USING THE SAME
Last renewal fee
Payment date Validity (years) Amount
2024-05-02 13 289.00 EUR
Legal status
Patent lapsed (non-payment of fees)
Invalidation date 2025-05-14