Herbas VPB

Print
EN | LT
LT - 1-((3-((1-Piperazinyl)carbonyl)phenyl)methyl)-2,4(1H,3H)-quinazolinedione derivatives as PARP inhibitors for treating cancer
EN - 1-((3-((1-Piperazinyl)carbonyl)phenyl)methyl)-2,4(1H,3H)-quinazolinedione derivatives as PARP inhibitors for treating cancer

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 239/96
C07D 401/06
A61K 31/517
A61P 9/00
A61P 35/00
European patent
(11) Number of the document 2709990
(13) Kind of document T
(96) European patent application number 12765230.3
Date of filing the European patent application 2012-03-31
(97) Date of publication of the European application 2014-03-26
(45) Date of publication and mention of the grant of the patent 2019-06-12
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/CN2012/073362
Date 2012-03-31
PCT application publication
(87) Number WO 2012/130166
Date 2012-10-04
Priority applications
(30) Number Date Country code
201110082475 2011-04-01 CN
PCT/CN2011/0770 2011-07-11 WO
Inventors
(72)
CAI, Sui Xiong, CN
TIAN, Ye Edward, CN
DONG, Haijun, CN
XU, Qingbing, CN
WU, Lizhen, CN
LIU, Lijun, CN
JIANG, Yangzhen, CN
BAO, Qingli, CN
WANG, Guoxiang, CN
YIN, Feng, CN
GU, Chengyun, CN
HU, Xiuhua, CN
WANG, Xiaozhu, CN
KANG, Sishun, CN
CHEN, Shengzhi, CN
Grantee
(73) Impact Therapeutics, Inc., Floor 9 10 Xinghuo Road Nanjing, Jiangsu 210061, CN
Title
(54) 1-((3-((1-Piperazinyl)carbonyl)phenyl)methyl)-2,4(1H,3H)-quinazolinedione derivatives as PARP inhibitors for treating cancer
  1-((3-((1-Piperazinyl)carbonyl)phenyl)methyl)-2,4(1H,3H)-quinazolinedione derivatives as PARP inhibitors for treating cancer