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LT - COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES
EN - COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 417/12
C07D 207/08
C07D 401/12
A61K 31/427
A61P 35/00
C07K 5/02
C07K 16/30
European patent
(11) Number of the document 2714684
(13) Kind of document T
(96) European patent application number 12793246.5
Date of filing the European patent application 2012-05-24
(97) Date of publication of the European application 2014-04-09
(45) Date of publication and mention of the grant of the patent 2018-09-05
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2012/039472
Date 2012-05-24
PCT application publication
(87) Number WO 2012/166560
Date 2012-12-06
Priority applications
(30) Number Date Country code
201161491146 P 2011-05-27 US
Inventors
(72)
MIAO, Zhenwei, US
ATKINSON, Kyle, C., US
BIROC, Sandra, US
BUSS, Timothy, US
COOK, Melissa, US
KRAYNOV, Vadim, US
MARSDEN, Robin, US
PINKSTAFF, Jason, US
SKIDMORE, Lillian, US
SUN, Ying, US
SZYDLIK, Angieszka, US
LOPEZ DE VALENTA, Delia Ianina, US
Grantee
(73) Ambrx, Inc., 10975 North Torrey Pines Road, Suite 100, La Jolla, CA 92037, US
Title
(54) COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES
  COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES