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LT - NOVEL METHOD FOR SYNTHESIZING RIVAROXABAN INTERMEDIATE, 4-{4-[(5S)-5-(AMINOMETHYL)-2-OXO-1,3-OXAZOLIDIN-3-YL]PHENYL}MORPHOLIN-3-ONE
EN - NOVEL METHOD FOR SYNTHESIZING RIVAROXABAN INTERMEDIATE, 4-{4-[(5S)-5-(AMINOMETHYL)-2-OXO-1,3-OXAZOLIDIN-3-YL]PHENYL}MORPHOLIN-3-ONE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 413/10
European patent
(11) Number of the document 2722330
(13) Kind of document T
(96) European patent application number 12799790.6
Date of filing the European patent application 2012-01-18
(97) Date of publication of the European application 2014-04-23
(45) Date of publication and mention of the grant of the patent 2017-04-26
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/CN2012/070530
Date 2012-01-18
PCT application publication
(87) Number WO 2012/171343
Date 2012-12-20
Priority applications
(30) Number Date Country code
201110158823 2011-06-14 CN
Inventors
(72)
ZI, Chunpeng, CN
HUANG, Luning, CN
ZHANG, Jeannie, CN
Grantee
(73) Zhejiang Huahai Pharmaceutical Co., Ltd, Xunqiao, Linhai, Zhejiang 317024, CN
Shanghai Syncores Technologies, Inc., 538 Cailun Rd Pudong, Shanghai 201203, CN
Title
(54) NOVEL METHOD FOR SYNTHESIZING RIVAROXABAN INTERMEDIATE, 4-{4-[(5S)-5-(AMINOMETHYL)-2-OXO-1,3-OXAZOLIDIN-3-YL]PHENYL}MORPHOLIN-3-ONE
  NOVEL METHOD FOR SYNTHESIZING RIVAROXABAN INTERMEDIATE, 4-{4-[(5S)-5-(AMINOMETHYL)-2-OXO-1,3-OXAZOLIDIN-3-YL]PHENYL}MORPHOLIN-3-ONE