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(51) | INT.CL. | C07D 413/10 |
(11) | Number of the document | 2722330 |
(13) | Kind of document | T |
(96) | European patent application number | 12799790.6 |
Date of filing the European patent application | 2012-01-18 | |
(97) | Date of publication of the European application | 2014-04-23 |
(45) | Date of publication and mention of the grant of the patent | 2017-04-26 |
(46) | Date of publication of the claims translation |
(86) | Number | PCT/CN2012/070530 |
Date | 2012-01-18 |
(87) | Number | WO 2012/171343 |
Date | 2012-12-20 |
(30) | Number | Date | Country code |
201110158823 | 2011-06-14 | CN |
(72) |
ZI, Chunpeng, CN
HUANG, Luning, CN
ZHANG, Jeannie, CN
|
(73) |
Zhejiang Huahai Pharmaceutical Co., Ltd,
Xunqiao, Linhai, Zhejiang 317024,
CN
Shanghai Syncores Technologies, Inc., 538 Cailun Rd Pudong, Shanghai 201203, CN |
(54) | NOVEL METHOD FOR SYNTHESIZING RIVAROXABAN INTERMEDIATE, 4-{4-[(5S)-5-(AMINOMETHYL)-2-OXO-1,3-OXAZOLIDIN-3-YL]PHENYL}MORPHOLIN-3-ONE |
NOVEL METHOD FOR SYNTHESIZING RIVAROXABAN INTERMEDIATE, 4-{4-[(5S)-5-(AMINOMETHYL)-2-OXO-1,3-OXAZOLIDIN-3-YL]PHENYL}MORPHOLIN-3-ONE |