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LT - PHARMACEUTICAL COMPOSITIONS OF 7-(6-(2-HYDROXYPROPAN-2-YL)PYRIDIN-3-YL)-1-((TRANS)-4-METHOXYCYCLOHEXYL)-3,4-DIHYDROPYRAZINO [2,3-B]PYRAZIN-2(1H)-ONE, A SOLID FORM THEREOF AND METHODS OF THEIR USE
EN - PHARMACEUTICAL COMPOSITIONS OF 7-(6-(2-HYDROXYPROPAN-2-YL)PYRIDIN-3-YL)-1-((TRANS)-4-METHOXYCYCLOHEXYL)-3,4-DIHYDROPYRAZINO [2,3-B]PYRAZIN-2(1H)-ONE, A SOLID FORM THEREOF AND METHODS OF THEIR USE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 9/00
A61K 9/20
A61K 9/28
A61K 31/4985
C07D 487/04
A61P 35/00
European patent
(11) Number of the document 2785325
(13) Kind of document T
(96) European patent application number 12798565.3
Date of filing the European patent application 2012-11-30
(97) Date of publication of the European application 2014-10-08
(45) Date of publication and mention of the grant of the patent 2018-08-22
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2012/067172
Date 2012-11-30
PCT application publication
(87) Number WO 2013/082344
Date 2013-06-06
Priority applications
(30) Number Date Country code
201161566109 P 2011-12-02 US
201261647288 P 2012-05-15 US
201261653439 P 2012-05-31 US
201261670419 P 2012-07-11 US
Inventors
(72)
CONNOLLY, Terrence, Joseph, US
KLOPFER, Kevin, Joseph, US
LEONG, William, Wei-Hwa, US
MENON, Anil, US
MIKLOS, Amanda, Nicole, US
KREILEIN, Matthew Michael, US
GAMBOA, Juan Antonio, US
XU, Jean, US
BOERSEN, Nathan, US
HUI, Ho-Wah, US
LEE, Thomas, CN
LI, Ying, US
COHEN, Benjamin, US
Grantee
(73) Signal Pharmaceuticals, LLC, 10300 Campus Point Drive, Suite 100, San Diego, CA 92121, US
Title
(54) PHARMACEUTICAL COMPOSITIONS OF 7-(6-(2-HYDROXYPROPAN-2-YL)PYRIDIN-3-YL)-1-((TRANS)-4-METHOXYCYCLOHEXYL)-3,4-DIHYDROPYRAZINO [2,3-B]PYRAZIN-2(1H)-ONE, A SOLID FORM THEREOF AND METHODS OF THEIR USE
  PHARMACEUTICAL COMPOSITIONS OF 7-(6-(2-HYDROXYPROPAN-2-YL)PYRIDIN-3-YL)-1-((TRANS)-4-METHOXYCYCLOHEXYL)-3,4-DIHYDROPYRAZINO [2,3-B]PYRAZIN-2(1H)-ONE, A SOLID FORM THEREOF AND METHODS OF THEIR USE