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LT - METHODS AND COMPOUNDS USEFUL IN THE SYNTHESIS OF OREXIN-2 RECEPTOR ANTAGONISTS
EN - METHODS AND COMPOUNDS USEFUL IN THE SYNTHESIS OF OREXIN-2 RECEPTOR ANTAGONISTS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07C 29/147
C07C 303/28
C07D 239/28
C12P 41/00
C07C 33/50
C07C 309/70
C07D 239/34
C07D 401/12
European patent
(11) Number of the document 2814798
(13) Kind of document T
(96) European patent application number 13706874.8
Date of filing the European patent application 2013-02-14
(97) Date of publication of the European application 2014-12-24
(45) Date of publication and mention of the grant of the patent 2019-04-03
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2013/026204
Date 2013-02-14
PCT application publication
(87) Number WO 2013/123240
Date 2013-08-22
Priority applications
(30) Number Date Country code
201261600109 P 2012-02-17 US
Inventors
(72)
MONIZ, George, Anthony, US
WILCOXEN, Annie, Zhu, US
BENAYOUD, Farid, US
LEE, Jaemoon, US
ZHANG, Huiming, US
TERAUCHI, Taro, JP
TAKEMURA, Ayumi, JP
YOSHIDA, Yu, JP
TANAKA, Toshiaki, JP
SORIMACHI, Keiichi, JP
NAOE, Yoshimitsu, JP
KAZUTA, Yuji, JP
Grantee
(73) Eisai R&D Management Co., Ltd., 6-10, Koishikawa 4-chome, Bunkyo-ku, Tokyo 112-8088, JP
Title
(54) METHODS AND COMPOUNDS USEFUL IN THE SYNTHESIS OF OREXIN-2 RECEPTOR ANTAGONISTS
  METHODS AND COMPOUNDS USEFUL IN THE SYNTHESIS OF OREXIN-2 RECEPTOR ANTAGONISTS