LT - ORAL SOLID DOSAGE FORMULATION OF 1,1-DIMETHYLETHYL [(1S)-1-{[(2S,4R)-4-(7-CHLORO-4METHOXYISOQUINOLIN-1-YLOXY)-2-({(1R,2S)-1-[(CYCLOPROPYLSULFONYL)CARBAMOYL]-2-ETHENYLCYCLOPROPYL}CARBAMOYL)PYRROLIDIN-1-YL]CARBONYL}-2,2-DIMETHYLPROPYL]CARBAMATE
EN - ORAL SOLID DOSAGE FORMULATION OF 1,1-DIMETHYLETHYL [(1S)-1-{[(2S,4R)-4-(7-CHLORO-4METHOXYISOQUINOLIN-1-YLOXY)-2-({(1R,2S)-1-[(CYCLOPROPYLSULFONYL)CARBAMOYL]-2-ETHENYLCYCLOPROPYL}CARBAMOYL)PYRROLIDIN-1-YL]CARBONYL}-2,2-DIMETHYLPROPYL]CARBAMATE
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
| (51) |
INT.CL. |
A61K 9/20 |
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A61K 31/4709 |
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A61P 31/14 |
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Europos patentas
| (11) |
Patento numeris |
2846778 |
| (13) |
Dokumento rūšis |
T |
| (96) |
Europos patento paraiškos numeris |
13722251.9 |
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Europos patento paraiškos padavimo data |
2013-05-03 |
| (97) |
Europos patento paraiškos paskelbimo data |
2015-03-18 |
| (45) |
Paskelbimo apie Europos patento išdavimą data |
2018-04-25
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| (46) |
Apibrėžties vertimo paskelbimo data |
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Tarptautinės paraiškos padavimo
| (86) |
Numeris |
PCT/US2013/039378 |
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Data |
2013-05-03 |
Tarptautinės paraiškos paskelbimo
| (87) |
Numeris |
WO 2013/169577 |
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Data |
2013-11-14 |
Prioriteto paraiškos
| (30) |
Numeris |
Data |
Šalis |
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201261643486 P |
2012-05-07
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US |
Išradėjai
| (72) |
HAMEY, Rhye, US
PANDEY, Preetanshu, US
BINDRA, Dilbir S., US
VEMAVARAPU, Chandra, US
PERRONE, Robert Kevin, US
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Savininkas
| (73) |
Bristol-Myers Squibb Holdings Ireland,
Hinterbergstrasse 16, Steinhausen,
CH
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Pavadinimas
| (54) |
ORAL SOLID DOSAGE FORMULATION OF 1,1-DIMETHYLETHYL [(1S)-1-{[(2S,4R)-4-(7-CHLORO-4METHOXYISOQUINOLIN-1-YLOXY)-2-({(1R,2S)-1-[(CYCLOPROPYLSULFONYL)CARBAMOYL]-2-ETHENYLCYCLOPROPYL}CARBAMOYL)PYRROLIDIN-1-YL]CARBONYL}-2,2-DIMETHYLPROPYL]CARBAMATE |
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ORAL SOLID DOSAGE FORMULATION OF 1,1-DIMETHYLETHYL [(1S)-1-{[(2S,4R)-4-(7-CHLORO-4METHOXYISOQUINOLIN-1-YLOXY)-2-({(1R,2S)-1-[(CYCLOPROPYLSULFONYL)CARBAMOYL]-2-ETHENYLCYCLOPROPYL}CARBAMOYL)PYRROLIDIN-1-YL]CARBONYL}-2,2-DIMETHYLPROPYL]CARBAMATE |