LT - NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS
EN - NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
(51) |
INT.CL. |
C07D 487/04 |
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A61K 31/4985 |
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A61P 3/10 |
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C07D 205/08 |
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European patent
(11) |
Number of the document |
2861598 |
(13) |
Kind of document |
T |
(96) |
European patent application number |
13730191.7 |
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Date of filing the European patent application |
2013-06-13 |
(97) |
Date of publication of the European application |
2015-04-22 |
(45) |
Date of publication and mention of the grant of the patent |
2017-10-25
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(46) |
Date of publication of the claims translation |
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PCT application
(86) |
Number |
PCT/EP2013/062307 |
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Date |
2013-06-13 |
PCT application publication
(87) |
Number |
WO 2013/186326 |
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Date |
2013-12-19 |
Priority applications
(30) |
Number |
Date |
Country code |
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12172012 |
2012-06-14
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EP |
Inventors
(72) |
STARCEVIC, Stefan, SI
MRAK, Peter, SI
KOPITAR, Gregor, SI
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Grantee
(73) |
LEK Pharmaceuticals d.d.,
Verovskova 57, 1526 Ljubljana,
SI
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Title
(54) |
NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS |
|
NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS |