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LT - NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS
EN - NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 487/04
A61K 31/4985
A61P 3/10
C07D 205/08
European patent
(11) Number of the document 2861598
(13) Kind of document T
(96) European patent application number 13730191.7
Date of filing the European patent application 2013-06-13
(97) Date of publication of the European application 2015-04-22
(45) Date of publication and mention of the grant of the patent 2017-10-25
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2013/062307
Date 2013-06-13
PCT application publication
(87) Number WO 2013/186326
Date 2013-12-19
Priority applications
(30) Number Date Country code
12172012 2012-06-14 EP
Inventors
(72)
STARCEVIC, Stefan, SI
MRAK, Peter, SI
KOPITAR, Gregor, SI
Grantee
(73) LEK Pharmaceuticals d.d., Verovskova 57, 1526 Ljubljana, SI
Title
(54) NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS
  NEW SYNTHETIC ROUTE FOR THE PREPARATION OF -AMINOBUTYRYL SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,4]DIAZOLO[4,3-a]PYRAZIN-7-YL COMPOUNDS