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LT - BENZIMIDAZOLE TETRAHYDROFURAN DERIVATIVES USEFUL AS AMP-ACTIVATED PROTEIN KINASE ACTIVATORS
EN - BENZIMIDAZOLE TETRAHYDROFURAN DERIVATIVES USEFUL AS AMP-ACTIVATED PROTEIN KINASE ACTIVATORS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 405/12
C07D 417/14
A61P 3/10
A61K 31/4184
A61K 31/415
A61K 31/454
European patent
(11) Number of the document 2888007
(13) Kind of document T
(96) European patent application number 13830944.8
Date of filing the European patent application 2013-08-15
(97) Date of publication of the European application 2015-07-01
(45) Date of publication and mention of the grant of the patent 2019-09-18
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2013/055166
Date 2013-08-15
PCT application publication
(87) Number WO 2014/031441
Date 2014-02-27
Priority applications
(30) Number Date Country code
201261692064 P 2012-08-22 US
Inventors
(72)
APGAR, James, M., US
BIFTU, Tesfaye, US
CHEN, Ping, US
FENG, Danqing, US
HICKS, Jacqueline, D., US
KEKEC, Ahmet, US
LEAVITT, Kenneth, J., US
LI, Bing, US
SEBHAT, Iyassu, US
QIAN, Xiaoxia, US
WEI, Lan, US
WILKENING, Robert, R., US
WU, Zhicai, US
Grantee
(73) Merck Sharp & Dohme Corp., 126 East Lincoln Avenue, Rahway, NJ 07065-0907, US
Title
(54) BENZIMIDAZOLE TETRAHYDROFURAN DERIVATIVES USEFUL AS AMP-ACTIVATED PROTEIN KINASE ACTIVATORS
  BENZIMIDAZOLE TETRAHYDROFURAN DERIVATIVES USEFUL AS AMP-ACTIVATED PROTEIN KINASE ACTIVATORS