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Teisinis statusas
Patentas galioja
(51) | INT.CL. | C07D 487/04 | (2006.01) |
A61K 31/495 | (2006.01) | ||
A61P 35/00 | (2006.01) |
(11) | Patento numeris | 2941432 |
(13) | Dokumento rūšis | T |
(96) | Europos patento paraiškos numeris | 13811716.3 |
Europos patento paraiškos padavimo data | 2013-12-06 | |
(97) | Europos patento paraiškos paskelbimo data | 2015-11-11 |
(45) | Paskelbimo apie Europos patento išdavimą data | 2018-03-07 |
(46) | Apibrėžties vertimo paskelbimo data | 2018-06-11 |
(86) | Numeris | PCT/US2013/073457 |
Data | 2013-12-06 |
(87) | Numeris | WO 2014/089379 |
Data | 2014-06-12 |
(30) | Numeris | Data | Šalis |
201261734726 P | 2012-12-07 | US | |
201361787568 P | 2013-03-15 | US | |
201361868132 P | 2013-08-21 | US |
(72) |
AHMAD, Nadia, GB
BOYALL, Dean, GB
CHARRIER, Jean-Damien, GB
DAVIS, Chris, GB
DAVIS, Rebecca, GB
DURRANT, Steven, GB
ETXEBARRIA I JARDI, Gorka, GB
FRAYSSE, Damien, GB
JIMENEZ, Juan-Miguel, GB
KAY, David, GB
KNEGTEL, Ronald, GB
MIDDLETON, Donald, GB
ODONNELL, Michael, GB
PANESAR, Maninder, GB
PIERARD, Francoise, GB
PINDER, Joanne, GB
SHAW, David, GB
STORCK, Pierre-Henri, GB
STUDLEY, John, GB
TWIN, Heather, GB
|
(73) |
Vertex Pharmaceuticals Incorporated,
50 Northern Avenue, Boston, MA 02210,
US
|
(74) |
Reda ŽABOLIENĖ,
METIDA, Verslo centras "VERTAS", Gynėjų g. 16, LT-01109 Vilnius,
LT
|
(54) | 2-Amino-6-fluor-N-(5-fluor-4-(4-(4-(oksetan-3-il)piperazin-1-karbonil)piperidin-1-il)piridin-3-il)pirazol[1,5alfa]pirimidin-3-karboksamidas kaip ATR kinazės inhibitorius |
2-AMINO-6-FLUORO-N-(5-FLUORO-4-(4-(4-(OXETAN-3-YL)PIPERAZINE-1-CARBONYL)PIPERIDIN-1-YL)PYRIDIN-3-YL)PYRAZOLO[1,5ALPHA]PYRIMIDINE-3-CARBOXAMIDE AS INHIBITOR OF ATR KINASE |
Mokėjimo data | Galiojimo metai | Suma | |
2024-11-19 | 12 | 289.00 EUR |
2025-12-06 |