LT - N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS
EN - N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
| (51) |
INT.CL. |
C07D 487/04 |
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A61K 31/4985 |
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A61P 25/00 |
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A61P 29/00 |
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Europos patentas
| (11) |
Patento numeris |
2978766 |
| (13) |
Dokumento rūšis |
T |
| (96) |
Europos patento paraiškos numeris |
14713845.7 |
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Europos patento paraiškos padavimo data |
2014-03-28 |
| (97) |
Europos patento paraiškos paskelbimo data |
2016-02-03 |
| (45) |
Paskelbimo apie Europos patento išdavimą data |
2018-12-19
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| (46) |
Apibrėžties vertimo paskelbimo data |
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Tarptautinės paraiškos padavimo
| (86) |
Numeris |
PCT/EP2014/056369 |
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Data |
2014-03-28 |
Tarptautinės paraiškos paskelbimo
| (87) |
Numeris |
WO 2014/154896 |
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Data |
2014-10-02 |
Prioriteto paraiškos
| (30) |
Numeris |
Data |
Šalis |
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13161864 |
2013-03-29
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EP |
Išradėjai
| (72) |
HOVEYDA, Hamid, BE
DUTHEUIL, Guillaume, BE
FRASER, Graeme, BE
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Savininkas
| (73) |
OGEDA SA,
Rue Adrienne Bolland, 47, 6041 Charleroi,
BE
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Pavadinimas
| (54) |
N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS |
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N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS |