LT - N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS
EN - N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) |
INT.CL. |
C07D 487/04 |
|
|
|
A61K 31/4985 |
|
|
|
A61P 25/00 |
|
|
|
A61P 29/00 |
|
Europos patentas
(11) |
Patento numeris |
2978766 |
(13) |
Dokumento rūšis |
T |
(96) |
Europos patento paraiškos numeris |
14713845.7 |
|
Europos patento paraiškos padavimo data |
2014-03-28 |
(97) |
Europos patento paraiškos paskelbimo data |
2016-02-03 |
(45) |
Paskelbimo apie Europos patento išdavimą data |
2018-12-19
|
(46) |
Apibrėžties vertimo paskelbimo data |
|
Tarptautinės paraiškos padavimo
(86) |
Numeris |
PCT/EP2014/056369 |
|
Data |
2014-03-28 |
Tarptautinės paraiškos paskelbimo
(87) |
Numeris |
WO 2014/154896 |
|
Data |
2014-10-02 |
Prioriteto paraiškos
(30) |
Numeris |
Data |
Šalis |
|
13161864 |
2013-03-29
|
EP |
Išradėjai
(72) |
HOVEYDA, Hamid, BE
DUTHEUIL, Guillaume, BE
FRASER, Graeme, BE
|
Savininkas
(73) |
OGEDA SA,
Rue Adrienne Bolland, 47, 6041 Charleroi,
BE
|
Pavadinimas
(54) |
N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS |
|
N-ACYL-(3-SUBSTITUTED)-5,6,7,8-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS |