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LT - 1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT
EN - 1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 47/68
C07D 487/04
C07D 209/60
A61P 35/00
C07K 16/00
C07K 16/28
C07K 16/30
C07K 16/32
C07D 207/40
C07D 209/62
C07D 401/12
C07D 401/14
C07D 403/14
C07D 471/04
C07H 15/24
European patent
(11) Number of the document 3033111
(13) Kind of document T
(96) European patent application number 14736243.8
Date of filing the European patent application 2014-06-16
(97) Date of publication of the European application 2016-06-22
(45) Date of publication and mention of the grant of the patent 2019-03-13
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2014/042560
Date 2014-06-16
PCT application publication
(87) Number WO 2015/023355
Date 2015-02-19
Priority applications
(30) Number Date Country code
201361864889 P 2013-08-12 US
201361916388 P 2013-12-16 US
201461969499 P 2014-03-24 US
Inventors
(72)
FLYGARE, John A., US
PILLOW, Thomas H., US
SAFINA, Brian, US
VERMA, Vishal, US
WEI, BinQing, US
DENNY, William, NZ
GIDDENS, Anna, NZ
LEE, Ho, NZ
LU, Guo-Liang, NZ
MILLER, Christian, NZ
REWCASTLE, Gordon, NZ
TERCEL, Moana, NZ
BONNET, Muriel, NZ
Grantee
(73) Genentech, Inc., 1 DNA Way, South San Francisco, CA 94080, US
Title
(54) 1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT
  1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT