LT - (2R)-4-okso-4-[3-(trifluormetil)-5,6- dihidro[L,2,4]triazolo[4,3-a]pirazin-7(8H)-il]-L-(2,4,5-trifluorfenil)butan-2-amino druskos su L-vyno rūgštimi stabilus polimorfas
EN - A STABLE POLYMORPH OF THE SALT OF (2R)-4-OXO-4-[3-(TRIFLUOROMETHYL)-5,6-DIHYDRO[L,2,4]TRIAZOLO[4,3-A]PYRAZIN-7(8H)-YL]-L-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE WITH L-TARTARIC ACID
Legal status
Patent lapsed (non-payment of fees)
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 487/04 |
(2006.01) |
|
|
C07C 59/255 |
(2006.01) |
European patent
| (11) |
Number of the document |
3063151 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
14815215.0 |
|
Date of filing the European patent application |
2014-10-30 |
| (97) |
Date of publication of the European application |
2016-09-07 |
| (45) |
Date of publication and mention of the grant of the patent |
2018-08-29
|
| (46) |
Date of publication of the claims translation |
2018-12-10
|
PCT application
| (86) |
Number |
PCT/CZ2014/000125 |
|
Date |
2014-10-30 |
PCT application publication
| (87) |
Number |
WO 2015/062562 |
|
Date |
2015-05-07 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
20130842 |
2013-11-01
|
CZ |
Inventors
| (72) |
RICHTER, Jindrich, CZ
LEHNERT, Petr, CZ
JARRAH, Kamal, CZ
DAMMER, Ondrej, CZ
KREJCIK, Lukas, CZ
|
Grantee
| (73) |
Zentiva K.S.,
U Kabelovny 130, 102 37 Praha 10,
CZ
|
Attorney or representative
| (74) |
Reda ŽABOLIENĖ,
METIDA, Verslo centras "VERTAS", Gynėjų g. 16, LT-01109 Vilnius,
LT
|
Title
| (54) |
(2R)-4-okso-4-[3-(trifluormetil)-5,6- dihidro[L,2,4]triazolo[4,3-a]pirazin-7(8H)-il]-L-(2,4,5-trifluorfenil)butan-2-amino druskos su L-vyno rūgštimi stabilus polimorfas |
| |
A STABLE POLYMORPH OF THE SALT OF (2R)-4-OXO-4-[3-(TRIFLUOROMETHYL)-5,6-DIHYDRO[L,2,4]TRIAZOLO[4,3-A]PYRAZIN-7(8H)-YL]-L-(2,4,5-TRIFLUOROPHENYL)BUTAN-2-AMINE WITH L-TARTARIC ACID |
Last renewal fee
|
Payment date |
Validity (years) |
Amount |
|
2020-09-16 |
7 |
162.00
EUR
|
Legal status
|
Patent lapsed (non-payment of fees)
|
|
|
Invalidation date |
2021-10-30 |
