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Legal status
Patent not validated
| (51) | INT.CL. | C07D 493/22 | |
| C07D 307/28 | |||
| C07C 6/02 |
| (11) | Number of the document | 3066102 |
| (13) | Kind of document | T |
| (96) | European patent application number | 14858240.6 |
| Date of filing the European patent application | 2014-11-04 | |
| (97) | Date of publication of the European application | 2016-09-14 |
| (45) | Date of publication and mention of the grant of the patent | 2020-02-26 |
| (46) | Date of publication of the claims translation |
| (86) | Number | PCT/US2014/063960 |
| Date | 2014-11-04 |
| (87) | Number | WO 2015/066729 |
| Date | 2015-05-07 |
| (30) | Number | Date | Country code |
| 201361899697 P | 2013-11-04 | US |
| (72) |
FANG, Francis, G., US
KIM, Dae-Shik, US
CHOI, Hyeong-Wook, US
CHASE, Charles, E., US
LEE, Jaemoon, US
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| (73) |
Eisai R&D Management Co., Ltd.,
6-10, Koishikawa 4-chome Bunkyo-ku, Tokyo 112-8088,
JP
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| (54) | MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B |
| MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B |