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LT - MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B
EN - MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 493/22
C07D 307/28
C07C 6/02
European patent
(11) Number of the document 3066102
(13) Kind of document T
(96) European patent application number 14858240.6
Date of filing the European patent application 2014-11-04
(97) Date of publication of the European application 2016-09-14
(45) Date of publication and mention of the grant of the patent 2020-02-26
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2014/063960
Date 2014-11-04
PCT application publication
(87) Number WO 2015/066729
Date 2015-05-07
Priority applications
(30) Number Date Country code
201361899697 P 2013-11-04 US
Inventors
(72)
FANG, Francis, G., US
KIM, Dae-Shik, US
CHOI, Hyeong-Wook, US
CHASE, Charles, E., US
LEE, Jaemoon, US
Grantee
(73) Eisai R&D Management Co., Ltd., 6-10, Koishikawa 4-chome Bunkyo-ku, Tokyo 112-8088, JP
Title
(54) MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B
  MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B