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LT - Kristalinė (S)-(2-(6-chlor-7-metil-1H-benzo[d]imidazol-2-il)-2-metilpirolidin-1-il)(5-metoksi-2-(2H-1,2,3-triazol-2-il)fenil)metanono forma ir jos panaudojimas kaip oreksino receptoriaus antagonisto
EN - CRYSTALLINE FORM OF (S)-(2-(6-CHLORO-7-METHYL-1H-BENZO[D]IMIDAZOL-2-YL)-2-METHYLPYRROLIDIN-1-YL)(5-METHOXY-2-(2H-1,2,3-TRIAZOL-2-YL)PHENYL)METHANONE AND ITS USE AS OREXIN RECEPTOR ANTAGONISTS

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Patent in force

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 403/14 (2006.01)
A61K 31/4192 (2006.01)
A61P 25/00 (2006.01)
European patent
(11) Number of the document 3077389
(13) Kind of document T
(96) European patent application number 14824107.8
Date of filing the European patent application 2014-12-02
(97) Date of publication of the European application 2016-10-12
(45) Date of publication and mention of the grant of the patent 2017-09-13
(46) Date of publication of the claims translation 2017-12-11
PCT application
(86) Number PCT/IB2014/066508
Date 2014-12-02
PCT application publication
(87) Number WO 2015/083070
Date 2015-06-11
Priority applications
(30) Number Date Country code
PCT/IB2013/0605 2013-12-03 WO
Inventors
(72)
BOSS, Christoph, CH
BROTSCHI, Christine, CH
GUDE, Markus, CH
HEIDMANN, Bibia, CH
SIFFERLEN, Thierry, CH
VON RAUMER, Markus, CH
WILLIAMS, Jodi, T., CH
Grantee
(73) Idorsia Pharmaceuticals Ltd, Hegenheimermattweg 91, 4123 Allschwil, CH
Attorney or representative
(74) Jurga PETNIŪNAITĖ, AAA Law, A. Goštauto g. 40B, Verslo centras "Dvyniai", LT-03163 Vilnius, LT
Title
(54) Kristalinė (S)-(2-(6-chlor-7-metil-1H-benzo[d]imidazol-2-il)-2-metilpirolidin-1-il)(5-metoksi-2-(2H-1,2,3-triazol-2-il)fenil)metanono forma ir jos panaudojimas kaip oreksino receptoriaus antagonisto
  CRYSTALLINE FORM OF (S)-(2-(6-CHLORO-7-METHYL-1H-BENZO[D]IMIDAZOL-2-YL)-2-METHYLPYRROLIDIN-1-YL)(5-METHOXY-2-(2H-1,2,3-TRIAZOL-2-YL)PHENYL)METHANONE AND ITS USE AS OREXIN RECEPTOR ANTAGONISTS
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2024-11-22 11 289.00 EUR
Next renewal fee
2025-12-02