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Legal status
Patent in force
| (51) | INT.CL. | C07D 487/04 | (2006.01) |
| C07B 59/00 | (2006.01) | ||
| A61K 31/519 | (2006.01) | ||
| A61P 35/00 | (2006.01) |
| (11) | Number of the document | 3077397 |
| (13) | Kind of document | T |
| (96) | European patent application number | 14815187.1 |
| Date of filing the European patent application | 2014-12-05 | |
| (97) | Date of publication of the European application | 2016-10-12 |
| (45) | Date of publication and mention of the grant of the patent | 2019-09-18 |
| (46) | Date of publication of the claims translation | 2020-01-27 |
| (86) | Number | PCT/US2014/068713 |
| Date | 2014-12-05 |
| (87) | Number | WO 2015/085132 |
| Date | 2015-06-11 |
| (30) | Number | Date | Country code |
| 201361912636 P | 2013-12-06 | US | |
| 201462008220 P | 2014-06-05 | US | |
| 201462058819 P | 2014-10-02 | US |
| (72) |
CHARRIER, Jean-Damien, GB
DAVIS, Christopher, John, GB
FRAYSSE, Damien, GB
ETXEBARRIA I JARDI, Gorka, GB
PEGG, Simon, GB
PIERARD, Francoise, GB
PINDER, Joanne, GB
STUDLEY, John, GB
ZWICKER, Carl, US
SANGHVI, Tapan, US
WALDO, Michael, US
MEDEK, Ales, US
SHAW, David, Matthew, GB
PANESAR, Maninder, GB
ZHANG, Yuegang, US
ALEM, Naziha, GB
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| (73) |
Vertex Pharmaceuticals Inc.,
50 Northern Avenue 15th Floor, Boston, MA 02210,
US
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| (74) |
Jurga PETNIŪNAITĖ,
AAA Law, A. Goštauto g. 40B, Verslo centras "Dvyniai", LT-03163 Vilnius,
LT
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| (54) | 2-Amino-6-fluor-N-[5-fluor-piridin-3-il]pirazolo[1,5-a]pirimidin-3-karboksamido junginys, naudingas kaip ATR kinazės inhibitorius, jo gamyba, skirtingos kietos formos ir jo radioaktyviai žymėti dariniai |
| 2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]PYRAZOLO[1,5-a]PYRIMIDIN-3-CARBOXAMIDE COMPOUND USEFUL AS ATR KINASE INHIBITOR, ITS PREPARATION, DIFFERENT SOLID FORMS AND RADIOLABELLED DERIVATIVES THEREOF |
| Payment date | Validity (years) | Amount | |
| 2025-11-18 | 12 | 289.00 EUR |
| 2026-12-05 |