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Legal status
Patent not validated
(51) | INT.CL. | A61K 47/68 | |
C07D 487/04 | |||
C07D 209/60 | |||
C07D 403/14 | |||
C07F 9/6558 | |||
C07F 9/6561 | |||
A61P 35/00 |
(11) | Number of the document | 3082876 |
(13) | Kind of document | T |
(96) | European patent application number | 14830914.9 |
Date of filing the European patent application | 2014-12-16 | |
(97) | Date of publication of the European application | 2016-10-26 |
(45) | Date of publication and mention of the grant of the patent | 2018-01-17 |
(46) | Date of publication of the claims translation |
(86) | Number | PCT/US2014/070637 |
Date | 2014-12-16 |
(87) | Number | WO 2015/095212 |
Date | 2015-06-25 |
(30) | Number | Date | Country code |
201361916388 P | 2013-12-16 | US | |
201461969499 P | 2014-03-24 | US | |
PCT/US2014/0425 | 2014-06-16 | WO |
(72) |
FLYGARE, John A., US
PILLOW, Thomas H., US
SAFINA, Brian, US
VERMA, Vishal, US
WEI, BinQing, US
DENNY, William, NZ
GIDDENS, Anna, NZ
LEE, Ho, NZ
LU, Guo-Liang, NZ
MILLER, Christian, NZ
REWCASTLE, Gordon, NZ
TERCEL, Moana, NZ
BONNET, Muriel, NZ
|
(73) |
Genentech, Inc.,
1 DNA Way, South San Francisco, CA 94080,
US
|
(54) | 1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT |
1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT |