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LT - 1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT
EN - 1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 47/68
C07D 487/04
C07D 209/60
C07D 403/14
C07F 9/6558
C07F 9/6561
A61P 35/00
European patent
(11) Number of the document 3082876
(13) Kind of document T
(96) European patent application number 14830914.9
Date of filing the European patent application 2014-12-16
(97) Date of publication of the European application 2016-10-26
(45) Date of publication and mention of the grant of the patent 2018-01-17
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2014/070637
Date 2014-12-16
PCT application publication
(87) Number WO 2015/095212
Date 2015-06-25
Priority applications
(30) Number Date Country code
201361916388 P 2013-12-16 US
201461969499 P 2014-03-24 US
PCT/US2014/0425 2014-06-16 WO
Inventors
(72)
FLYGARE, John A., US
PILLOW, Thomas H., US
SAFINA, Brian, US
VERMA, Vishal, US
WEI, BinQing, US
DENNY, William, NZ
GIDDENS, Anna, NZ
LEE, Ho, NZ
LU, Guo-Liang, NZ
MILLER, Christian, NZ
REWCASTLE, Gordon, NZ
TERCEL, Moana, NZ
BONNET, Muriel, NZ
Grantee
(73) Genentech, Inc., 1 DNA Way, South San Francisco, CA 94080, US
Title
(54) 1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT
  1-(CHLOROMETHYL)-2,3-DIHYDRO-1H-BENZO[E]INDOLE DIMER ANTIBODY-DRUG CONJUGATE COMPOUNDS, AND METHODS OF USE AND TREATMENT