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Legal status
Patent not validated
| (51) | INT.CL. | C07D 471/20 | (2006.01) |
| A61K 31/499 | (2013.01) | ||
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| C07D 495/20 | (2006.01) | ||
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| A61K 31/427 | (2006.01) | ||
| A61K 31/675 | (2013.01) | ||
| A61K 31/499 | (2006.01) | ||
| C07D 475/10 | (2013.01) | ||
| A61K 31/513 | (2006.01) | ||
| C07D 491/10 | (2013.01) | ||
| A61K 31/52 | (2006.01) | ||
| C07D 495/10 | (2013.01) | ||
| A61K 31/53 | (2006.01) | ||
| A61K 31/53 | (2013.01) | ||
| A61K 31/55 | (2006.01) | ||
| C07D 491/20 | (2013.01) | ||
| A61K 31/675 | (2006.01) | ||
| C07D 495/20 | (2013.01) | ||
| A61P 31/18 | (2006.01) | ||
| A61P 31/18 | (2018.01) |
| (11) | Number of the document | 3083641 |
| (13) | Kind of document | T |
| (96) | European patent application number | 14870755.7 |
| Date of filing the European patent application | 2014-12-17 | |
| (97) | Date of publication of the European application | 2016-10-26 |
| (45) | Date of publication and mention of the grant of the patent | 2022-11-09 |
| (46) | Date of publication of the claims translation |
| (86) | Number | PCT/US2014/070712 |
| Date | 2014-12-17 |
| (87) | Number | WO 2015/095258 |
| Date | 2015-06-25 |
| (30) | Number | Date | Country code |
| PCT/CN2013/090156 | 2013-12-20 | WO |
| (72) |
GRAHAM, Thomas, H. , US
LIU, Wensheng , US
YU, Tao , US
ZHANG, Yonglian , US
WADDELL, Sherman, T. , US
WAI, John, S. , US
COLEMAN, Paul, J. , US
SANDERS, John, M. , US
EMBREY, Mark, W. , US
WALJI, Abbas, M. , US
FERGUSON, Ronald Dale, II , US
DI MARCO, Christina Ng , US
STEELE, Thomas, G. , US
HU, Lihong , CN
PENG, Xuanjia , CN
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| (73) |
Merck Sharp & Dohme LLC ,
126 East Lincoln Avenue, Rahway, New Jersey 07065-0907,
US
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| (54) | SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS |
| SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS |