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LT - SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS
EN - SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 471/20 (2006.01)
A61K 31/499 (2013.01)
C07D 471/22 (2006.01)
A61K 31/55 (2013.01)
C07D 471/20 (2013.01)
C07D 475/10 (2006.01)
C07D 471/22 (2013.01)
C07D 491/10 (2006.01)
C07D 491/20 (2006.01)
A61K 31/427 (2013.01)
C07D 495/10 (2006.01)
A61K 31/513 (2013.01)
C07D 495/20 (2006.01)
A61K 31/52 (2013.01)
A61K 31/427 (2006.01)
A61K 31/675 (2013.01)
A61K 31/499 (2006.01)
C07D 475/10 (2013.01)
A61K 31/513 (2006.01)
C07D 491/10 (2013.01)
A61K 31/52 (2006.01)
C07D 495/10 (2013.01)
A61K 31/53 (2006.01)
A61K 31/53 (2013.01)
A61K 31/55 (2006.01)
C07D 491/20 (2013.01)
A61K 31/675 (2006.01)
C07D 495/20 (2013.01)
A61P 31/18 (2006.01)
A61P 31/18 (2018.01)
European patent
(11) Number of the document 3083641
(13) Kind of document T
(96) European patent application number 14870755.7
Date of filing the European patent application 2014-12-17
(97) Date of publication of the European application 2016-10-26
(45) Date of publication and mention of the grant of the patent 2022-11-09
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2014/070712
Date 2014-12-17
PCT application publication
(87) Number WO 2015/095258
Date 2015-06-25
Priority applications
(30) Number Date Country code
PCT/CN2013/090156 2013-12-20 WO
Inventors
(72)
GRAHAM, Thomas, H. , US
LIU, Wensheng , US
YU, Tao , US
ZHANG, Yonglian , US
WADDELL, Sherman, T. , US
WAI, John, S. , US
COLEMAN, Paul, J. , US
SANDERS, John, M. , US
EMBREY, Mark, W. , US
WALJI, Abbas, M. , US
FERGUSON, Ronald Dale, II , US
DI MARCO, Christina Ng , US
STEELE, Thomas, G. , US
HU, Lihong , CN
PENG, Xuanjia , CN
Grantee
(73) Merck Sharp & Dohme LLC , 126 East Lincoln Avenue, Rahway, New Jersey 07065-0907, US
Title
(54) SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS
  SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS