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LT - DEUTERATED HETEROCYCLE FUSED GAMMA-CARBOLINES AS ANTAGONISTS OF 5-HT2A RECEPTORS
EN - DEUTERATED HETEROCYCLE FUSED GAMMA-CARBOLINES AS ANTAGONISTS OF 5-HT2A RECEPTORS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/4985 (2006.01)
C07D 471/14 (2013.01)
C07D 471/14 (2006.01)
A61K 45/06 (2013.01)
C07B 59/002 (2013.01)
A61K 45/06 (2006.01)
A61K 31/4985 (2013.01)
C07D 471/16 (2006.01)
A61P 25/00 (2006.01)
C07D 471/16 (2013.01)
C07B 59/00 (2006.01)
A61P 1/00 (2018.01)
A61P 1/00 (2006.01)
A61P 21/02 (2018.01)
A61P 3/04 (2006.01)
A61P 25/00 (2018.01)
A61P 21/02 (2006.01)
A61P 25/04 (2018.01)
A61P 25/14 (2018.01)
A61P 25/04 (2006.01)
A61P 25/16 (2018.01)
A61P 25/14 (2006.01)
A61P 25/18 (2018.01)
A61P 25/16 (2006.01)
A61P 25/18 (2006.01)
A61P 25/20 (2018.01)
A61P 25/20 (2006.01)
A61P 25/22 (2018.01)
A61P 25/22 (2006.01)
A61P 25/24 (2018.01)
A61P 25/24 (2006.01)
A61P 25/28 (2018.01)
A61P 29/02 (2006.01)
A61P 29/02 (2018.01)
A61P 43/00 (2006.01)
A61P 3/04 (2018.01)
A61P 25/28 (2006.01)
A61P 43/00 (2018.01)
European patent
(11) Number of the document 3125893
(13) Kind of document T
(96) European patent application number 15773589.5
Date of filing the European patent application 2015-04-03
(97) Date of publication of the European application 2017-02-08
(45) Date of publication and mention of the grant of the patent 2023-09-20
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2015/024340
Date 2015-04-03
PCT application publication
(87) Number WO 2015/154025
Date 2015-10-08
Priority applications
(30) Number Date Country code
201461975610 P 2014-04-04 US
Inventors
(72)
MATES, Sharon , US
LI, Peng , US
WENNOGLE, Lawrence P. , US
DAVIS, Robert , US
Grantee
(73) Intra-Cellular Therapies, Inc. , 430 East 29th Street, Suite 900, New York, NY 10016, US
Title
(54) DEUTERATED HETEROCYCLE FUSED GAMMA-CARBOLINES AS ANTAGONISTS OF 5-HT2A RECEPTORS
  DEUTERATED HETEROCYCLE FUSED GAMMA-CARBOLINES AS ANTAGONISTS OF 5-HT2A RECEPTORS