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Legal status
Patent not validated
(51) | INT.CL. | A61K 31/42 | (2006.01) |
A61P 9/00 | (2006.01) | ||
C07D 261/00 | (2006.01) | ||
C07D 413/14 | (2006.01) | ||
A61K 45/06 | (2006.01) | ||
A61K 31/397 | (2006.01) | ||
A61K 31/4245 | (2006.01) | ||
A61K 31/4439 | (2006.01) | ||
A61K 31/444 | (2006.01) | ||
C07D 413/10 | (2006.01) | ||
C07D 261/04 | (2006.01) |
(11) | Number of the document | 3174537 |
(13) | Kind of document | T |
(96) | European patent application number | 15827553.7 |
Date of filing the European patent application | 2015-07-24 | |
(97) | Date of publication of the European application | 2017-06-07 |
(45) | Date of publication and mention of the grant of the patent | 2021-06-23 |
(46) | Date of publication of the claims translation |
(86) | Number | PCT/US2015/041871 |
Date | 2015-07-24 |
(87) | Number | WO 2016/018729 |
Date | 2016-02-04 |
(30) | Number | Date | Country code |
201462030229 P | 2014-07-29 | US |
(72) |
SHAO, Pengcheng Patrick , US
YE, Feng , US
VACHAL, Petr , US
THATAI, Jayanth Thiruvellore , IN
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(73) |
Merck Sharp & Dohme Corp. ,
126 East Lincoln Avenue, Rahway, NJ 07065-0907,
US
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(54) | MONOCYCLIC ISOXAZOLINES AS INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN |
MONOCYCLIC ISOXAZOLINES AS INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN |