Herbas VPB

Print
EN | LT
LT - MONOCYCLIC ISOXAZOLINES AS INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN
EN - MONOCYCLIC ISOXAZOLINES AS INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/42 (2006.01)
A61P 9/00 (2006.01)
C07D 261/00 (2006.01)
C07D 413/14 (2006.01)
A61K 45/06 (2006.01)
A61K 31/397 (2006.01)
A61K 31/4245 (2006.01)
A61K 31/4439 (2006.01)
A61K 31/444 (2006.01)
C07D 413/10 (2006.01)
C07D 261/04 (2006.01)
European patent
(11) Number of the document 3174537
(13) Kind of document T
(96) European patent application number 15827553.7
Date of filing the European patent application 2015-07-24
(97) Date of publication of the European application 2017-06-07
(45) Date of publication and mention of the grant of the patent 2021-06-23
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2015/041871
Date 2015-07-24
PCT application publication
(87) Number WO 2016/018729
Date 2016-02-04
Priority applications
(30) Number Date Country code
201462030229 P 2014-07-29 US
Inventors
(72)
SHAO, Pengcheng Patrick , US
YE, Feng , US
VACHAL, Petr , US
THATAI, Jayanth Thiruvellore , IN
Grantee
(73) Merck Sharp & Dohme Corp. , 126 East Lincoln Avenue, Rahway, NJ 07065-0907, US
Title
(54) MONOCYCLIC ISOXAZOLINES AS INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN
  MONOCYCLIC ISOXAZOLINES AS INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN