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EN | LT
LT - SYNTHETIC INTERMEDIATE OF (R)-1(2,2 -DIFLUOROBENZO[D][1,3]DIOXOL-5YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2YL)-1H-INDOL-5YL)CYCLOPROPANECARBOXAMIDE
EN - SYNTHETIC INTERMEDIATE OF (R)-1(2,2 -DIFLUOROBENZO[D][1,3]DIOXOL-5YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2YL)-1H-INDOL-5YL)CYCLOPROPANECARBOXAMIDE

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 405/12 (2006.01)
Europos patentas
(11) Patento numeris 3181561
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 17154840.7
Europos patento paraiškos padavimo data 2011-03-25
(97) Europos patento paraiškos paskelbimo data 2017-06-21
(45) Paskelbimo apie Europos patento išdavimą data 2020-05-20
(46) Apibrėžties vertimo paskelbimo data
Prioriteto paraiškos
(30) Numeris Data Šalis
317376 P 2010-03-25 US
319953 P 2010-04-01 US
321636 P 2010-04-07 US
321561 P 2010-04-07 US
Išradėjai
(72)
Keshavarz-Shokri, Ali, US
Zhang, Beili, US
Alcacio, Tim Edward, US
Lee, Elaine Chungmin, US
Zhang, Yuegang, US
Krawiec, Mariusz, US
Nugent, William A., US
Savininkas
(73) Vertex Pharmaceuticals Incorporated, 50 Northern Avenue, Boston, MA 02210, US
Pavadinimas
(54) SYNTHETIC INTERMEDIATE OF (R)-1(2,2 -DIFLUOROBENZO[D][1,3]DIOXOL-5YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2YL)-1H-INDOL-5YL)CYCLOPROPANECARBOXAMIDE
  SYNTHETIC INTERMEDIATE OF (R)-1(2,2 -DIFLUOROBENZO[D][1,3]DIOXOL-5YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2YL)-1H-INDOL-5YL)CYCLOPROPANECARBOXAMIDE