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LT - NOVEL SALTS OF 3-[(DIMETHYLAMINO)METHYL]-N-{2-[4-(HYDROXYCARBAMOYL) PHENOXY]ETHYL}-1-BENZOFURAN-2-CARBOXAMIDE, RELATED CRYSTALLINE FORMS, METHOD FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
EN - NOVEL SALTS OF 3-[(DIMETHYLAMINO)METHYL]-N-{2-[4-(HYDROXYCARBAMOYL) PHENOXY]ETHYL}-1-BENZOFURAN-2-CARBOXAMIDE, RELATED CRYSTALLINE FORMS, METHOD FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 307/85
A61K 31/343
A61P 35/00
European patent
(11) Number of the document 3189040
(13) Kind of document T
(96) European patent application number 15767627.1
Date of filing the European patent application 2015-09-03
(97) Date of publication of the European application 2017-07-12
(45) Date of publication and mention of the grant of the patent 2020-07-29
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2015/048243
Date 2015-09-03
PCT application publication
(87) Number WO 2016/036910
Date 2016-03-10
Priority applications
(30) Number Date Country code
1458224 2014-09-03 FR
1458215 2014-09-03 FR
Inventors
(72)
GAILLARD, Marina, FR
LETELLIER, Philippe, FR
Grantee
(73) Pharmacyclics LLC, 995 East Arques Avenue, Sunnyvale, CA 94085, US
Title
(54) NOVEL SALTS OF 3-[(DIMETHYLAMINO)METHYL]-N-{2-[4-(HYDROXYCARBAMOYL) PHENOXY]ETHYL}-1-BENZOFURAN-2-CARBOXAMIDE, RELATED CRYSTALLINE FORMS, METHOD FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
  NOVEL SALTS OF 3-[(DIMETHYLAMINO)METHYL]-N-{2-[4-(HYDROXYCARBAMOYL) PHENOXY]ETHYL}-1-BENZOFURAN-2-CARBOXAMIDE, RELATED CRYSTALLINE FORMS, METHOD FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME