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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
| (51) | INT.CL. | C07D 471/04 | (2006.01) |
| A61P 11/00 | (2018.01) | ||
| C07D 519/00 | (2006.01) | ||
| A61P 25/16 | (2018.01) | ||
| A61K 31/437 | (2006.01) | ||
| A61P 43/00 | (2018.01) | ||
| A61K 31/553 | (2006.01) | ||
| A61P 17/16 | (2018.01) | ||
| A61P 25/00 | (2018.01) | ||
| A61P 29/00 | (2006.01) | ||
| A61P 37/00 | (2006.01) | ||
| A61P 5/14 | (2018.01) | ||
| A61P 1/16 | (2018.01) | ||
| A61P 29/00 | (2018.01) | ||
| A61P 3/10 | (2018.01) | ||
| A61P 11/02 | (2018.01) | ||
| A61P 1/04 | (2018.01) | ||
| A61P 25/28 | (2018.01) | ||
| A61P 17/00 | (2018.01) | ||
| A61P 19/02 | (2018.01) | ||
| A61P 21/00 | (2018.01) | ||
| A61P 7/04 | (2018.01) | ||
| A61P 11/06 | (2018.01) | ||
| A61P 1/02 | (2018.01) | ||
| A61P 19/00 | (2018.01) | ||
| A61P 9/10 | (2018.01) | ||
| A61P 9/00 | (2018.01) | ||
| A61P 37/08 | (2018.01) | ||
| A61P 37/02 | (2018.01) | ||
| A61P 5/38 | (2018.01) | ||
| A61P 7/06 | (2018.01) | ||
| C07D 471/04 | (2013.01) | ||
| C07D 519/00 | (2013.01) | ||
| A61P 17/06 | (2018.01) | ||
| A61P 1/18 | (2018.01) | ||
| A61P 13/02 | (2018.01) | ||
| A61P 37/00 | (2018.01) | ||
| A61P 37/06 | (2018.01) | ||
| A61P 21/04 | (2018.01) | ||
| A61P 13/12 | (2018.01) | ||
| A61P 31/04 | (2018.01) | ||
| A61P 17/14 | (2018.01) | ||
| A61P 7/00 | (2018.01) |
| (11) | Patento numeris | 3204382 |
| (13) | Dokumento rūšis | T |
| (96) | Europos patento paraiškos numeris | 15784212.1 |
| Europos patento paraiškos padavimo data | 2015-10-06 | |
| (97) | Europos patento paraiškos paskelbimo data | 2017-08-16 |
| (45) | Paskelbimo apie Europos patento išdavimą data | 2021-12-01 |
| (46) | Apibrėžties vertimo paskelbimo data |
| (86) | Numeris | PCT/US2015/054221 |
| Data | 2015-10-06 |
| (87) | Numeris | WO 2016/057500 |
| Data | 2016-04-14 |
| (30) | Numeris | Data | Šalis |
| 201462060249 P | 2014-10-06 | US |
| (72) |
GAILLARD, Pascale , FR
SEENISAMY, Jeyaprakashnarayanan , IN
LIU-BUJALSKI, Lesley , US
POTNICK, Justin , US
CALDWELL, Richard D. , US
QIU, Hui , US
NEAGU, Constantin , US
JONES, Reinaldo , US
WON, Annie Cho , US
GOUTOPOULOS, Andreas , US
SHERER, Brian A. , US
JOHNSON, Theresa L. , US
GARDBERG, Anna , US
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| (73) |
Merck Patent GmbH ,
Frankfurter Strasse 250, 64293 Darmstadt,
DE
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| (54) | HETEROARYL COMPOUNDS AS BTK INHIBITORS AND USES THEREOF |
| HETEROARYL COMPOUNDS AS BTK INHIBITORS AND USES THEREOF |