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LT - SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS
EN - SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/499 (2006.01)
A61K 31/499 (2013.01)
A61P 31/18 (2006.01)
A61K 45/06 (2013.01)
A61K 31/675 (2006.01)
A61P 31/18 (2018.01)
A61K 31/683 (2006.01)
C07D 491/20 (2013.01)
C07D 487/20 (2006.01)
A61K 31/675 (2013.01)
C07D 491/20 (2006.01)
A61K 31/683 (2013.01)
C07F 9/6561 (2006.01)
C07D 487/20 (2013.01)
A61K 45/06 (2006.01)
C07F 9/6561 (2013.01)
European patent
(11) Number of the document 3229805
(13) Kind of document T
(96) European patent application number 15868594.1
Date of filing the European patent application 2015-12-04
(97) Date of publication of the European application 2017-10-18
(45) Date of publication and mention of the grant of the patent 2023-04-19
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2015/063850
Date 2015-12-04
PCT application publication
(87) Number WO 2016/094197
Date 2016-06-16
Priority applications
(30) Number Date Country code
PCT/CN2014/093335 2014-12-09 WO
Inventors
(72)
EMBREY, Mark, W. , US
GRAHAM, Thomas, H. , US
RAHEEM, Izzat, T. , US
SCHREIER, John, D. , US
WADDELL, Sherman, T. , US
WAI, John, S. , US
HU, Lihong , CN
PENG, Xuanjia , CN
Grantee
(73) Merck Sharp & Dohme LLC , 126 East Lincoln Avenue, Rahway, New Jersey 07065, US
Title
(54) SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS
  SPIROCYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS