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LT - PROCESS FOR THE PREPARATION OF (3Z,5S)-5-(HYDROXYMETHYL)-1-[(2´-METHYL-1,1´-BIPHENYL-4-YL)CARBONYL)PYRROLIDIN-3-ONE O-METHYLOXIME
EN - PROCESS FOR THE PREPARATION OF (3Z,5S)-5-(HYDROXYMETHYL)-1-[(2´-METHYL-1,1´-BIPHENYL-4-YL)CARBONYL)PYRROLIDIN-3-ONE O-METHYLOXIME

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 207/09 (2013.01)
C07D 207/22 (2006.01)
A61K 31/4025 (2006.01)
C07D 207/22 (2013.01)
A61P 5/10 (2006.01)
A61K 31/40 (2013.01)
A61P 13/08 (2018.01)
A61P 15/00 (2018.01)
A61P 15/04 (2018.01)
A61P 15/06 (2018.01)
A61P 15/08 (2018.01)
A61P 15/10 (2018.01)
A61P 25/00 (2018.01)
A61P 25/02 (2018.01)
A61P 25/14 (2018.01)
A61P 25/18 (2018.01)
A61P 25/22 (2018.01)
A61P 25/24 (2018.01)
A61P 3/14 (2018.01)
A61P 43/00 (2018.01)
A61P 5/00 (2018.01)
A61P 5/10 (2018.01)
A61P 5/38 (2018.01)
A61P 5/40 (2018.01)
A61P 9/00 (2018.01)
A61P 9/08 (2018.01)
European patent
(11) Number of the document 3252037
(13) Kind of document T
(96) European patent application number 17177956.4
Date of filing the European patent application 2014-07-25
(97) Date of publication of the European application 2017-12-06
(45) Date of publication and mention of the grant of the patent 2022-03-09
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
13183723 2013-09-10 EP
Inventors
(72)
CHOLLET, André , CH
Grantee
(73) ObsEva S.A. , 12, Chemin des Aulx, 1228 Plan-les-Ouates/Geneve, CH
Title
(54) PROCESS FOR THE PREPARATION OF (3Z,5S)-5-(HYDROXYMETHYL)-1-[(2´-METHYL-1,1´-BIPHENYL-4-YL)CARBONYL)PYRROLIDIN-3-ONE O-METHYLOXIME
  PROCESS FOR THE PREPARATION OF (3Z,5S)-5-(HYDROXYMETHYL)-1-[(2´-METHYL-1,1´-BIPHENYL-4-YL)CARBONYL)PYRROLIDIN-3-ONE O-METHYLOXIME